SCHEMBL30372136

SCHEMBL30372136

CN(C)S(=O)(=O)c1ccccc1Nc1nc(Nc2ccc(N3CCOCC3)cc2)nc2[nH]ccc12

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 6/20 0.66
TTK P33981 5/20 0.61
PTK2 Q05397 7/20 0.57
AXL P30530 1/20 0.57
NEK2 P51955 1/20 0.57
JAK2 O60674 1/20 0.52
BRD4 O60885 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29017307 1.00 MAP4K1 (0.66) MAP4K1TTKPTK2AXLNEK2
SCHEMBL30372758 0.91 AXL (0.69) MAP4K1TTKPTK2AXLNEK2
SCHEMBL29017290 0.89 TTK (0.65) MAP4K1TTKPTK2
SCHEMBL30372090 0.89 EGFR (0.59) MAP4K1TTKPTK2AXLNEK2
SCHEMBL29017297 0.80 AXL (0.58) MAP4K1TTKPTK2AXLNEK2
SCHEMBL30372483 0.80 AXL (0.58) MAP4K1TTKPTK2AXLNEK2
SCHEMBL30372722 0.80 MAP4K1 (0.81) MAP4K1AXLNEK2
SCHEMBL29017414 0.80 MAP4K1 (0.81) MAP4K1AXLNEK2
SCHEMBL14547750 0.78 TTK (0.63) TTKPTK2JAK2
SCHEMBL23566970 0.77 EGFR (0.77) TTKPTK2JAK2BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116239597-B Pyrimidine pyrrole derivative and medicinal composition and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-116239597-A Pyrimidine pyrrole derivative and medicinal composition and application thereof 中国科学院上海药物研究所 2023-06-09 CN disclosed