SCHEMBL30385474

SCHEMBL30385474

COC(=O)c1cc(F)c(Br)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.46
LCK P06239 1/20 0.44
MAPT P10636 3/20 0.42
GABRP O00591 2/20 0.42
GABRD O14764 2/20 0.42
GABRA1 P14867 2/20 0.42
GABRB1 P18505 2/20 0.42
GABRG2 P18507 2/20 0.42
GABRB3 P28472 2/20 0.42
GABRA5 P31644 2/20 0.42
GABRA3 P34903 2/20 0.42
GABRA2 P47869 2/20 0.42
GABRB2 P47870 2/20 0.42
GABRA4 P48169 2/20 0.42
GABRE P78334 2/20 0.42
GABRA6 Q16445 2/20 0.42
GABRG1 Q8N1C3 2/20 0.42
GABRG3 Q99928 2/20 0.42
GABRQ Q9UN88 2/20 0.42
KDM4E B2RXH2 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17130053 1.00 MAPK1 (0.46) MAPK1LCKMAPTGABRPGABRD
SCHEMBL21652771 0.86 MAPK1 (0.46) MAPK1LCKMAPTGABRPGABRD
SCHEMBL1459953 0.81 MAPK1 (0.47) MAPK1LCKMAPTGABRPGABRD
SCHEMBL23611991 0.81 LCK (0.53) MAPK1LCKMAPTGABRPGABRD
SCHEMBL9400422 0.81 MAPK1 (0.47) MAPK1LCKMAPTGABRPGABRD
SCHEMBL16318862 0.79 MAPK1 (0.46) MAPK1LCKMAPTGABRPGABRD
SCHEMBL18340557 0.79 MAPK1 (0.46) MAPK1LCKMAPTGABRPGABRD
SCHEMBL29260500 0.79 MAPK1 (0.46) MAPK1LCKMAPTGABRPGABRD
SCHEMBL23481999 0.79 MAPK1 (0.50) MAPK1LCKMAPTGABRPGABRD
SCHEMBL31435378 0.79 NOTUM (0.55) MAPK1LCKMAPTGABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115919859-B Pharmaceutical composition of heteroaryl derivative and application of pharmaceutical composition in medicine 四川海思科制药有限公司 2024-01-05 CN disclosed
CN-115919859-A Pharmaceutical composition of heteroaryl derivative and application thereof in medicine 四川海思科制药有限公司 2023-04-07 CN disclosed