SCHEMBL30401798

SCHEMBL30401798

COc1ccc(CNc2ncnc3c(C(=O)Nc4c(C)ccc5c(Nc6cc(F)c(F)cc6F)nccc45)cccc23)c(OC)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKA O14965 13/20 0.49
RPS6KB1 P23443 7/20 0.49
AURKB Q96GD4 8/20 0.47
RAF1 P04049 5/20 0.45
BRAF P15056 5/20 0.45
MAPT P10636 1/20 0.44
CSF1R P07333 2/20 0.43
DDR1 Q08345 2/20 0.43
DDR2 Q16832 2/20 0.43
ARAF P10398 1/20 0.43
ALDH1A1 P00352 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25374976 1.00 AURKA (0.49) AURKARPS6KB1AURKBRAF1BRAF
SCHEMBL30401863 0.95 AURKA (0.49) AURKARPS6KB1AURKBRAF1BRAF
SCHEMBL30402488 0.95 AURKA (0.49) AURKARPS6KB1AURKBRAF1BRAF
SCHEMBL24399693 0.95 AURKA (0.49) AURKARPS6KB1AURKBRAF1BRAF
SCHEMBL24399606 0.95 AURKA (0.49) AURKARPS6KB1AURKBRAF1BRAF
SCHEMBL25376015 0.93 AURKA (0.48) AURKARPS6KB1AURKBRAF1BRAF
SCHEMBL25372766 0.93 AURKA (0.48) AURKARPS6KB1AURKBRAF1BRAF
SCHEMBL24399562 0.93 AURKA (0.48) AURKARPS6KB1AURKBRAF1BRAF
SCHEMBL25375423 0.93 AURKA (0.48) AURKARPS6KB1AURKBRAF1BRAF
SCHEMBL30401799 0.93 AURKA (0.48) AURKARPS6KB1AURKBRAF1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116096718-A Aryl amide compound, pharmaceutical composition containing same, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2023-05-09 CN disclosed