SCHEMBL30409556

SCHEMBL30409556

Cc1nnc(-c2ccc3[nH]ncc3c2)o1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.55
CDK2 P24941 2/20 0.55
CCNE1 P24864 1/20 0.55
DBF4 Q9UBU7 1/20 0.55
TRPA1 O75762 7/20 0.52
GSK3B P49841 5/20 0.51
CLK1 P49759 2/20 0.51
CDK5 Q00535 2/20 0.51
DYRK1A Q13627 2/20 0.51
DYRK3 O43781 1/20 0.51
CLK2 P49760 1/20 0.51
CLK3 P49761 1/20 0.51
CDK5R1 Q15078 1/20 0.51
DYRK2 Q92630 1/20 0.51
CLK4 Q9HAZ1 1/20 0.51
DYRK1B Q9Y463 1/20 0.51
ROCK2 O75116 3/20 0.50
PIM1 P11309 3/20 0.50
AURKB Q96GD4 3/20 0.50
S1PR1 P21453 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25185033 1.00 CDC7 (0.55) CDC7CDK2CCNE1DBF4TRPA1
SCHEMBL3490816 0.82 CDC7 (0.55) CDC7CDK2CCNE1DBF4TRPA1
SCHEMBL2191369 0.78 CDK2 (0.71) CDC7CDK2CCNE1DBF4TRPA1
SCHEMBL2191428 0.74 GSK3B (0.53) CDC7CDK2CCNE1DBF4TRPA1
SCHEMBL16573980 0.74 GSK3B (0.71) CDK2TRPA1GSK3BCLK1CDK5
SCHEMBL23558460 0.73 CDC7 (0.45) CDC7CDK2CCNE1DBF4TRPA1
SCHEMBL13963952 0.73 NPC1 (0.47) PIM1LRRK2
SCHEMBL25195476 0.73 TLR8 (0.46) CDC7CDK2CCNE1DBF4GSK3B
SCHEMBL13332229 0.73 S1PR1 (0.60) CDK2TRPA1GSK3BCLK1CDK5
SCHEMBL6984735 0.72 SMN1; SMN2 (0.73)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023078337-A1 CDK8/19 DUAL INHIBITORS AND METHODS OF USE INSILICO MEDICINE IP LIMITED (CN) 2023-05-11 WO disclosed