SCHEMBL30413445

SCHEMBL30413445

Nc1nnc(-c2c3ccccc3cc3ccccc23)c(N)n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK1A1 P48729 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
MGAM O43451 1/20 0.47
GAA P10253 1/20 0.47
SI P14410 1/20 0.47
MGAM2 Q2M2H8 1/20 0.47
ADORA2A P29274 8/20 0.43
ADORA1 P30542 8/20 0.43
CYP2D6 P10635 1/20 0.42
MAOA P21397 1/20 0.42
MAPK1 P28482 1/20 0.42
ADRA1A P35348 1/20 0.42
SCN4A P35499 1/20 0.42
BLM P54132 1/20 0.42
PMP22 Q01453 1/20 0.42
PDE3A Q14432 1/20 0.42
SCN5A Q14524 1/20 0.42
SCN9A Q15858 1/20 0.42
SCN2A Q99250 1/20 0.42
SCN3A Q9NY46 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL979602 1.00 CSNK1A1 (0.55) CSNK1A1CLK4MGAMGAASI
SCHEMBL748850 0.81 CSNK1A1 (0.50) CSNK1A1CLK4ADORA2AADORA1CYP2D6
SCHEMBL3702933 0.79 CYP2D6 (0.51) CSNK1A1CLK4MGAMGAASI
SCHEMBL17350861 0.77 CSNK1A1 (0.45) CSNK1A1CLK4MGAMGAASI
SCHEMBL6374321 0.76 CSNK1A1 (0.47) CSNK1A1CLK4ADORA2AADORA1CYP2D6
SCHEMBL978392 0.75 CYP2D6 (0.58) CSNK1A1CLK4ADORA2AADORA1CYP2D6
SCHEMBL17350868 0.72 ADORA2A (0.50) CSNK1A1CLK4ADORA2AADORA1CYP2D6
SCHEMBL976510 0.71 ADORA2A (0.71) CSNK1A1CLK4ADORA2AADORA1KDM4E
SCHEMBL976667 0.71 CSNK1A1 (1.00) CSNK1A1CLK4GAAADORA2AADORA1
SCHEMBL976598 0.70 SCN9A (0.67) CSNK1A1CLK4ADORA2AADORA1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002280-B1 CYCLIC TRIAZO AND DIAZO SODIUM CHANNEL BLOCKERS UNIV GREENWICH (GB) 2023-05-24 EP disclosed