SCHEMBL30414738

SCHEMBL30414738

CCc1cnc2cc(CN3CCN(c4ccc(OC(F)F)nc4)CC3)cnc2c1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.72
PARP2 Q9UGN5 8/20 0.72
PARP6 Q2NL67 3/20 0.45
PARP3 Q9Y6F1 3/20 0.45
TNKS O95271 1/20 0.45
TIPARP Q7Z3E1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30414526 0.88 PARP1 (0.58) PARP1PARP2PARP6PARP3TNKS
SCHEMBL25192086 0.84 PARP1 (1.00) PARP1PARP2PARP6PARP3TNKS
SCHEMBL30893600 0.80 PARP1 (0.49) PARP1PARP2PARP6PARP3TNKS
SCHEMBL31424725 0.79 PARP1 (0.55) PARP1PARP2PARP6PARP3TNKS
SCHEMBL30414803 0.79 PARP1 (0.49) PARP1PARP2
SCHEMBL30893591 0.77 PARP1 (0.52) PARP1PARP2PARP6PARP3TNKS
SCHEMBL20962645 0.75 PARP1 (0.51) PARP1PARP2
SCHEMBL30414229 0.75 PARP1 (0.48) PARP1PARP2PARP6PARP3TNKS
SCHEMBL30385483 0.74 PARP1 (0.50) PARP1PARP2PARP6PARP3TNKS
SCHEMBL30385332 0.74 PARP1 (0.52) PARP1PARP2PARP6PARP3TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118055933-A Selective PARP1 inhibitors and uses thereof 成都百裕制药股份有限公司 2024-05-17 CN disclosed
WO-2023088408-A1 SELECTIVE PARP1 INHIBITOR AND APPLICATION THEREOF 成都百裕制药股份有限公司 2023-05-25 WO disclosed