SCHEMBL30424940

SCHEMBL30424940

CC(C)(C)OC(=O)Nc1cc2cc(N3CCN(C4(C)COCC4F)CC3)c(Cl)cc2cn1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 18/20 0.58
KCNH2 Q12809 7/20 0.47
BRSK1 Q8TDC3 1/20 0.47
MARK3 P27448 1/20 0.45
SCN5A Q14524 1/20 0.45
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29567817 1.00 LRRK2 (0.58) LRRK2KCNH2BRSK1MARK3SCN5A
SCHEMBL24394351 1.00 LRRK2 (0.58) LRRK2KCNH2BRSK1MARK3SCN5A
SCHEMBL29568017 0.87 LRRK2 (0.48) LRRK2KCNH2BRSK1MARK3SCN5A
SCHEMBL24394350 0.87 LRRK2 (0.48) LRRK2KCNH2BRSK1MARK3SCN5A
SCHEMBL30424449 0.87 LRRK2 (0.48) LRRK2KCNH2BRSK1MARK3SCN5A
SCHEMBL29568377 0.85 LRRK2 (0.78) LRRK2KCNH2BRSK1MARK3SCN5A
SCHEMBL29567993 0.85 LRRK2 (0.78) LRRK2KCNH2BRSK1MARK3SCN5A
SCHEMBL29567808 0.85 LRRK2 (0.78) LRRK2KCNH2BRSK1MARK3SCN5A
SCHEMBL29567756 0.85 LRRK2 (0.78) LRRK2KCNH2BRSK1MARK3SCN5A
SCHEMBL26965839 0.85 LRRK2 (0.78) LRRK2KCNH2BRSK1MARK3SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116390727-A N-linked isoquinolinamides as LRRK2 inhibitors, pharmaceutical compositions and uses thereof 默沙东有限责任公司 2023-07-04 CN disclosed