SCHEMBL30425571

SCHEMBL30425571

CC(C)(C)OC(=O)N1CCc2cccc(Nc3nc(Cl)ncc3Cl)c21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNK O75909 1/20 0.49
CCNA2 P20248 1/20 0.49
CDK2 P24941 1/20 0.49
CCND3 P30281 1/20 0.49
CDK9 P50750 1/20 0.49
CDK6 Q00534 1/20 0.49
ALK Q9UM73 6/20 0.44
STK17B O94768 1/20 0.41
STK17A Q9UEE5 1/20 0.41
EGFR P00533 3/20 0.40
NOTUM Q6P988 1/20 0.39
MAP4K1 Q92918 2/20 0.38
MAP3K7 O43318 4/20 0.38
MAPK1 P28482 2/20 0.38
MAP2K1 Q02750 2/20 0.38
INSR P06213 2/20 0.37
FGFR1 P11362 1/20 0.37
SRC P12931 1/20 0.37
SLC2A1 P11166 1/20 0.37
MET P08581 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26655582 1.00 CCNK (0.49) CCNKCCNA2CDK2CCND3CDK9
SCHEMBL25004485 0.86 NOTUM (0.55) ALKEGFRNOTUMMAP3K7MAPK1
SCHEMBL25005396 0.83 MAP3K7 (0.44) CCNKCCNA2CDK2CCND3CDK9
SCHEMBL25005398 0.80 NOTUM (0.47) ALKEGFRNOTUMMAP3K7MAPK1
SCHEMBL29114931 0.79 EGFR (0.43) CCNKCCNA2CDK2CCND3CDK9
SCHEMBL25005397 0.78 MAP3K7 (0.43) ALKEGFRMAP3K7MAPK1MAP2K1
SCHEMBL30425857 0.76 ALK (0.70) CDK2ALKSTK17BSTK17AEGFR
SCHEMBL26655424 0.76 ALK (0.70) CDK2ALKSTK17BSTK17AEGFR
SCHEMBL31147629 0.76 NOTUM (0.50) ALKNOTUM
SCHEMBL27237971 0.76 NOTUM (0.50) ALKNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116249690-A Indoline compounds and derivatives as EGFR inhibitors 百济神州有限公司 2023-06-09 CN disclosed