SCHEMBL30434855

SCHEMBL30434855

COc1cccc2nc(-c3cc(C)c(OCCO)c(C)c3)[nH]c(=O)c12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 13/20 0.61
PARP1 P09874 2/20 0.61
HDAC1 Q13547 5/20 0.56
IL17A Q16552 1/20 0.55
HDAC3 O15379 3/20 0.55
HDAC4 P56524 3/20 0.55
HDAC7 Q8WUI4 3/20 0.55
HDAC2 Q92769 3/20 0.55
HDAC10 Q969S8 3/20 0.55
HDAC11 Q96DB2 3/20 0.55
HDAC8 Q9BY41 3/20 0.55
HDAC6 Q9UBN7 3/20 0.55
HDAC9 Q9UKV0 3/20 0.55
HDAC5 Q9UQL6 3/20 0.55
BRD1 O95696 1/20 0.45
BRD2 P25440 1/20 0.45
MMP13 P45452 1/20 0.43
CYP1A1 P04798 2/20 0.43
CYP1B1 Q16678 2/20 0.43
GUSB P08236 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL149925 1.00 BRD4 (0.61) BRD4PARP1HDAC1IL17AHDAC3
SCHEMBL377714 0.91 BRD4 (0.57) BRD4PARP1HDAC1IL17AHDAC3
SCHEMBL15551676 0.88 BRD4 (0.54) BRD4PARP1HDAC1IL17AHDAC3
SCHEMBL25694623 0.86 BRD4 (0.69) BRD4PARP1HDAC1IL17AHDAC3
SCHEMBL122791 0.86 PBRM1 (0.60) BRD4PARP1HDAC1IL17AHDAC3
SCHEMBL30434926 0.86 PBRM1 (0.60) BRD4PARP1HDAC1IL17AHDAC3
SCHEMBL378245 0.85 BRD4 (0.77) BRD4PARP1HDAC1IL17AHDAC3
Apabetalone SCHEMBL29352238 0.85 BRD4 (0.84) BRD4PARP1HDAC1IL17AHDAC3
Apabetalone SCHEMBL145019 0.85 BRD4 (0.84) BRD4PARP1HDAC1IL17AHDAC3
SCHEMBL143261 0.84 BRD4 (0.66) BRD4PARP1HDAC1IL17AHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107252429-B Novel anti-inflammatory agent 雷斯韦洛吉克斯公司 2023-06-16 CN disclosed