SCHEMBL30445112

SCHEMBL30445112

Cc1cc(-n2cc(C=O)nn2)ncc1C#N

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 19/20 0.40
KCNH2 Q12809 1/20 0.40
P2RX7 Q99572 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20168342 1.00 KCNJ1 (0.40) KCNJ1KCNH2P2RX7
SCHEMBL30445053 0.83 KCNJ1 (0.45) KCNJ1P2RX7
SCHEMBL20168352 0.83 KCNJ1 (0.45) KCNJ1P2RX7
SCHEMBL30444275 0.80 KCNJ1 (0.40) KCNJ1KCNH2P2RX7
SCHEMBL20574919 0.80 KCNJ1 (0.40) KCNJ1KCNH2P2RX7
SCHEMBL30445023 0.80 KCNJ1 (0.44) KCNJ1KCNH2
SCHEMBL20168545 0.80 KCNJ1 (0.44) KCNJ1KCNH2
SCHEMBL20574979 0.78 KCNJ1 (0.42) KCNJ1KCNH2
SCHEMBL20575137 0.78 KCNJ1 (0.42) KCNJ1KCNH2
SCHEMBL30444323 0.78 KCNJ1 (0.42) KCNJ1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110139862-B Substituted bicyclic heterocyclic derivatives useful as ROMK channel inhibitors 百时美施贵宝公司 2024-01-16 CN disclosed
CN-110678463-B Substituted nitrogen-containing compounds 百时美施贵宝公司 2023-06-06 CN disclosed