SCHEMBL30445161

SCHEMBL30445161

COc1nc(-n2cc(CO)nn2)cc(C)c1C#N

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 4/20 0.51
RECQL P46063 1/20 0.47
NOTUM Q6P988 11/20 0.45
P2RX7 Q99572 1/20 0.43
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20176989 1.00 KCNJ1 (0.51) KCNJ1RECQLNOTUMP2RX7POLB
SCHEMBL30445299 0.85 KCNJ1 (0.49) KCNJ1NOTUMP2RX7L3MBTL1IRAK4
SCHEMBL20168069 0.85 KCNJ1 (0.49) KCNJ1NOTUMP2RX7L3MBTL1IRAK4
SCHEMBL30445081 0.81 KCNJ1 (0.48) KCNJ1NOTUMP2RX7MAPK1
SCHEMBL20575090 0.81 KCNJ1 (0.48) KCNJ1NOTUMP2RX7MAPK1
SCHEMBL20168469 0.80 RECQL (0.48) KCNJ1RECQLP2RX7POLBTSHR
SCHEMBL30444334 0.80 RECQL (0.48) KCNJ1RECQLP2RX7POLBTSHR
SCHEMBL2592972 0.78 RECQL (0.61) RECQLPOLBTSHRMAPK1
SCHEMBL20176988 0.76 RECQL (0.47) KCNJ1RECQLP2RX7POLBTSHR
SCHEMBL30445572 0.76 RECQL (0.47) KCNJ1RECQLP2RX7POLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110139862-B Substituted bicyclic heterocyclic derivatives useful as ROMK channel inhibitors 百时美施贵宝公司 2024-01-16 CN disclosed
CN-110678463-B Substituted nitrogen-containing compounds 百时美施贵宝公司 2023-06-06 CN disclosed