SCHEMBL30453738

SCHEMBL30453738

CNS(=O)(=O)c1ccc(OC)c(Nc2ncc(F)c(N(C)c3ccc4c(C)n[nH]c4c3)n2)c1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 11/20 0.41
BRAF P15056 6/20 0.38
PARP1 P09874 1/20 0.36
KDR P35968 1/20 0.36
PAK1 Q13153 1/20 0.36
MAP2K4 P45985 1/20 0.36
GAK O14976 1/20 0.35
LRRK2 Q5S007 1/20 0.34
ZAP70 P43403 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL589246 1.00 TNNI3K (0.41) TNNI3KBRAFPARP1KDRPAK1
SCHEMBL588579 0.92 KDR (0.36) TNNI3KPARP1KDRPAK1MAP2K4
SCHEMBL31672566 0.92 KDR (0.41) PARP1KDRPAK1
SCHEMBL10151145 0.92 KDR (0.41) PARP1KDRPAK1
SCHEMBL31672412 0.90 ALK (0.39) PARP1KDRPAK1
SCHEMBL2877867 0.90 ALK (0.39) PARP1KDRPAK1
SCHEMBL30453279 0.85 LRRK2 (0.38) KDRPAK1LRRK2
SCHEMBL589240 0.85 LRRK2 (0.38) KDRPAK1LRRK2
SCHEMBL589264 0.85 KDR (0.46) TNNI3KBRAFPARP1KDRMAP2K4
SCHEMBL30453307 0.85 KDR (0.46) TNNI3KBRAFPARP1KDRMAP2K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113181362-B Medicament for preventing and/or treating amyotrophic lateral sclerosis 国立大学法人京都大学 2023-06-13 CN disclosed