SCHEMBL30454154

SCHEMBL30454154

Cc1n[nH]c2cc(N(C)c3nc(Nc4cccc(S(=O)(=O)NC(C)C)c4)ncc3F)ccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
KDR P35968 3/20 0.43
BRD4 O60885 6/20 0.42
PAK1 Q13153 2/20 0.41
CDK2 P24941 5/20 0.40
CCNT1 O60563 4/20 0.40
CDK1 P06493 4/20 0.40
CCNB1 P14635 4/20 0.40
CDK9 P50750 4/20 0.40
CCNA2 P20248 3/20 0.40
CDK7 P50613 3/20 0.40
CCNH P51946 3/20 0.40
CCNE2 O96020 3/20 0.40
CCNE1 P24864 3/20 0.40
CCNB2 O95067 2/20 0.40
CCNB3 Q8WWL7 2/20 0.40
CCNA1 P78396 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL589319 1.00 CYP3A4 (0.43) CYP3A4CYP2D6CYP2C9CYP2C19KDR
SCHEMBL31672454 0.85 PAK1 (0.42) CYP3A4CYP2D6CYP2C9CYP2C19KDR
SCHEMBL2867774 0.85 PAK1 (0.42) CYP3A4CYP2D6CYP2C9CYP2C19KDR
SCHEMBL588579 0.85 KDR (0.36) KDRPAK1MAP2K4
SCHEMBL589173 0.85 KDR (0.60) CYP3A4CYP2D6CYP2C9CYP2C19KDR
SCHEMBL31672441 0.84 KDR (0.46) CYP3A4CYP2D6CYP2C9CYP2C19KDR
SCHEMBL2877133 0.84 KDR (0.46) CYP3A4CYP2D6CYP2C9CYP2C19KDR
SCHEMBL2873675 0.82 PAK1 (0.48) CYP3A4CYP2D6CYP2C9CYP2C19KDR
SCHEMBL31672493 0.82 PAK1 (0.48) CYP3A4CYP2D6CYP2C9CYP2C19KDR
SCHEMBL589261 0.82 CDK2 (0.44) CYP3A4CYP2D6CYP2C9CYP2C19KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113181362-B Medicament for preventing and/or treating amyotrophic lateral sclerosis 国立大学法人京都大学 2023-06-13 CN disclosed