SCHEMBL30456324

SCHEMBL30456324

CP(C)(=O)c1c(C(=O)O)ccc2c(-c3nc(N[C@H]4CC[C@H](NCCOCCN)C4)ncc3C(F)(F)F)c[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCNK O75909 16/20 0.49
CDK12 Q9NYV4 16/20 0.49
CCNT1 O60563 15/20 0.49
CCNE1 P24864 15/20 0.49
CDK2 P24941 15/20 0.49
CDK9 P50750 15/20 0.49
CDK7 P50613 12/20 0.49
CCNH P51946 12/20 0.49
MNAT1 P51948 9/20 0.49
CYP2D6 P10635 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25363678 1.00 CCNK (0.49) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL31220711 0.92 CCNK (0.51) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL25363014 0.92 CCNK (0.51) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL31220745 0.91 CCNK (0.51) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL25360542 0.91 CCNK (0.51) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL25363261 0.91 CCNK (0.50) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL31220678 0.91 CCNK (0.50) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL31220649 0.91 CCNK (0.47) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL31220662 0.89 CCNK (0.50) CCNKCDK12CCNT1CCNE1CDK2
SCHEMBL25363464 0.89 CCNK (0.50) CCNKCDK12CCNT1CCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4455132-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE Insilico Medicine IP Limited (HK) 2024-10-30 EP disclosed
WO-2023116761-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE 英矽智能科技知识产权有限公司 2023-06-29 WO disclosed