SCHEMBL30459502

SCHEMBL30459502

O=C(O)N1CCC(Nc2ncc3ccc(=O)n(C4CCCC4)c3n2)CC1

nearest known ligand 0.71

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 17/20 0.71
CCND1 P24385 17/20 0.71
CCNE1 P24864 16/20 0.71
CDK6 Q00534 14/20 0.71
CDK4 P11802 7/20 0.71
CCNT1 O60563 3/20 0.71
CDK9 P50750 3/20 0.71
MAPK8 P45983 1/20 0.66
MAPK9 P45984 1/20 0.66
MAPK10 P53779 1/20 0.66
CCND3 P30281 4/20 0.60
CCND2 P30279 3/20 0.60
FGFR1 P11362 1/20 0.60
CCNA2 P20248 1/20 0.60
FGFR2 P21802 1/20 0.60
FGFR4 P22455 1/20 0.60
FGFR3 P22607 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3303713 0.95 CCND1 (0.66) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL16802783 0.87 MAPK8 (0.76) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL5269917 0.86 CCND1 (0.78) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL3306096 0.86 CCND1 (0.78) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL24572106 0.85 CCNE1 (0.66) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL30459572 0.85 CCNE1 (0.66) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL16802795 0.84 CDK2 (0.74) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL18148251 0.84 CDK2 (0.74) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL26098322 0.84 CCNE1 (0.61) CDK2CCND1CCNE1CDK6CDK4
SCHEMBL26098323 0.84 CCNE1 (0.61) CDK2CCND1CCNE1CDK6CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023051302-A1 HETEROCYCLIC COMPOUND HAVING CYCLIN-DEPENDENT KINASE INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 中国医药研究开发中心有限公司 2023-04-06 WO disclosed