SCHEMBL30459766

SCHEMBL30459766

C=CC(=O)Nc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.68
EPHX2 P34913 3/20 0.67
TEK Q02763 2/20 0.63
TGM2 P21980 7/20 0.63
EPHB4 P54760 1/20 0.60
MAPT P10636 1/20 0.57
TRPV1 Q8NER1 2/20 0.55
F13A1 P00488 1/20 0.54
LMNA P02545 1/20 0.54
TGM1 P22735 1/20 0.54
TGM3 Q08188 1/20 0.54
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA9 Q16790 1/20 0.53
FAAH O00519 1/20 0.52
ALDH1A1 P00352 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27767000 0.84 KMT2A (0.69) KMT2AEPHX2TEKEPHB4MAPT
SCHEMBL18812119 0.83 MAPT (0.61) KMT2AEPHX2TEKEPHB4MAPT
SCHEMBL29277130 0.81 EGFR (0.65) EPHX2TEKTGM2EPHB4MAPT
SCHEMBL30684939 0.81 EGFR (0.65) EPHX2TEKTGM2EPHB4MAPT
SCHEMBL9285859 0.81 KMT2A (0.64) KMT2AEPHX2MAPTTRPV1CA12
SCHEMBL2090980 0.81 KMT2A (0.64) KMT2AEPHX2MAPTTRPV1LMNA
SCHEMBL8858788 0.81 KMT2A (0.73) KMT2AEPHX2MAPTTRPV1LMNA
SCHEMBL9265165 0.81 KMT2A (0.64) KMT2AEPHX2MAPTTRPV1CA12
SCHEMBL8858784 0.81 KMT2A (0.73) KMT2AEPHX2MAPTTRPV1LMNA
SCHEMBL11555827 0.80 EPHX2 (1.00) KMT2AEPHX2MAPTTRPV1FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117069700-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-11-17 CN disclosed
CN-111170999-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-06-30 CN disclosed