SCHEMBL30459783

SCHEMBL30459783

COc1ccc(Nc2ccnc(Cl)n2)c(N)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.47
EGFR P00533 3/20 0.46
GAA P10253 3/20 0.44
MAPT P10636 4/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
LMNA P02545 2/20 0.43
ALDH1A1 P00352 2/20 0.43
NPC1 O15118 1/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 1/20 0.43
NOS3 P29474 1/20 0.41
NOS1 P29475 1/20 0.41
NOS2 P35228 1/20 0.41
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LCK P06239 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17683162 1.00 ROCK1 (0.47) ROCK1EGFRGAAMAPTMEN1
SCHEMBL4820325 0.85 GAA (0.62) EGFRGAAMAPTMEN1KMT2A
SCHEMBL21676903 0.84 ROCK1 (0.47) ROCK1EGFRGAAMAPTMEN1
SCHEMBL30108000 0.82 MAPT (0.53) EGFRGAAMAPTMEN1KMT2A
SCHEMBL3638254 0.82 LCK (0.56) ROCK1EGFRGAAMAPTMEN1
SCHEMBL18386919 0.82 APP (0.40) ROCK1MEN1KMT2ANOS3NOS1
SCHEMBL20632859 0.82 ROCK1 (0.45) ROCK1EGFRGAAMAPTMEN1
SCHEMBL30010939 0.81 ROCK1 (0.46) ROCK1ALDH1A1MAPK1SMN1; SMN2PIK3CA
SCHEMBL20162211 0.81 ROCK1 (0.46) ROCK1ALDH1A1MAPK1SMN1; SMN2PIK3CA
SCHEMBL4433403 0.81 MEN1 (0.43) ROCK1EGFRGAAMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402143-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2024-01-16 CN disclosed
CN-117069700-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-11-17 CN disclosed
CN-111187221-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-26 CN disclosed
CN-111171000-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-01 CN disclosed
CN-111170999-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-06-30 CN disclosed