SCHEMBL30468418

SCHEMBL30468418

CC(C)(C)OC(=O)N1CCc2ccc(Nc3ncc(C(F)(F)F)c(Cl)n3)cc2C1

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 16/20 0.55
FLT3 P36888 16/20 0.55
KIT P10721 6/20 0.55
MAPT P10636 1/20 0.54
IGF1R P08069 1/20 0.51
NR1H2 P55055 1/20 0.49
JAK2 O60674 1/20 0.49
JAK3 P52333 1/20 0.49
PTK2 Q05397 1/20 0.49
MAP3K7 O43318 1/20 0.49
RPS6KB1 P23443 1/20 0.49
PRKAG1 P54619 1/20 0.49
PRKAA2 P54646 1/20 0.49
KCNH2 Q12809 1/20 0.49
PRKAB1 Q9Y478 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29051888 1.00 CHEK1 (0.55) CHEK1FLT3KITMAPTIGF1R
SCHEMBL23754874 0.96 CHEK1 (0.57) CHEK1FLT3KITMAPTJAK2
SCHEMBL30088400 0.96 CHEK1 (0.57) CHEK1FLT3KITMAPTJAK2
SCHEMBL30468449 0.93 CHEK1 (0.52) CHEK1FLT3KITMAPTMAP3K7
SCHEMBL23764769 0.93 CHEK1 (0.52) CHEK1FLT3KITMAPTMAP3K7
SCHEMBL4283268 0.87 MAPT (0.50) CHEK1FLT3KITMAPTIGF1R
SCHEMBL25234686 0.86 TYRO3 (0.59) CHEK1FLT3KIT
SCHEMBL30412224 0.86 TYRO3 (0.59) CHEK1FLT3KIT
SCHEMBL23764827 0.86 CHEK1 (0.75) CHEK1FLT3KITMAP3K7RPS6KB1
SCHEMBL30741470 0.86 CHEK1 (0.75) CHEK1FLT3KITMAP3K7RPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332910-A 2-aminopyrimidine derivatives as kinase inhibitors, preparation and use thereof 江苏威凯尔医药科技有限公司 2023-06-27 CN disclosed