Guanidine

Guanidine

SCHEMBL3047699

COS(=O)(=O)O.N=C(N)N

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3

The experimentally established mechanism targets of Guanidine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
BLM P54132 2/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C19 P33261 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CA2 P00918 3/20 0.42
CA1 P00915 2/20 0.42
TSHR P16473 3/20 0.37
USP2 O75604 1/20 0.37
NT5E P21589 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
F2 P00734 2/20 0.32
PRSS1 P07477 2/20 0.32
PRSS2 P07478 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetamidine SCHEMBL6287555 0.91 BLM (0.43) KDM4EBLMCYP2D6CYP2C19NPSR1
Thiourea SCHEMBL7362564 0.88 KDM4E (0.42) KDM4EBLMCYP2D6CYP2C19NPSR1
SCHEMBL6737394 0.88 KDM4E (0.42) KDM4EBLMCYP2D6CYP2C19NPSR1
SCHEMBL6286669 0.84 KDM4E (0.39) KDM4EBLMCYP2D6CYP2C19NPSR1
SCHEMBL6289391 0.84 KDM4E (0.39) KDM4EBLMCYP2D6CYP2C19NPSR1
Hydrazine SCHEMBL679587 0.83
Methylamine SCHEMBL143865 0.83
Hydroxyamine SCHEMBL27900806 0.83
SCHEMBL27308161 0.83 TSHR (0.50) KDM4ECA2CA1TSHRUSP2
SCHEMBL5991 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118240806-A Liquid thrombin reagent 仪器实验室公司 2024-06-25 CN disclosed
CN-114072378-B Process (III) for preparing metastable crystal modifications of N- (aminoiminomethyl) -2-glycine 澳泽化学特罗斯特贝格有限公司 2024-02-02 CN disclosed
CN-109566664-A A kind of aquatic products, livestock and poultry disinfectant and its preparation and application 南京瑞碧斯生物科技有限公司 2019-04-05 CN disclosed
US-20100222580-A1 Process For The Preparation Of Onium Alkylsulfates Having A Low Halide Content MERCK PATENT GMBH (DE) 2010-09-02 US disclosed
EP-1828142-B1 METHOD FOR PRODUCING ONIUM ALKYL SULFATES WITH A LOW HALOGENIDE CONTENT MERCK PATENT GMBH (DE) 2010-06-02 EP disclosed
EP-1828142-A1 METHOD FOR PRODUCING ONIUM ALKYL SULFATES WITH A LOW HALOGENIDE CONTENT Merck Patent GmbH (DE) 2007-09-05 EP disclosed
CN-1301978-C Preparation of 2-methyl-4-pyrimidone LUYUAN PHARMACEUTICAL CO LTD D (CN) 2007-02-28 CN disclosed
WO-2006063654-A1 METHOD FOR PRODUCING ONIUM ALKYL SULFATES WITH A LOW HALOGENIDE CONTENT MERCK PATENT GMBH (DE) 2006-06-22 WO disclosed
CN-1491939-A Hexa alkyl guanidine salt ion liquid and preparing process 中国科学院长春应用化学研究所 2004-04-28 CN disclosed
US-5635322-A Process for developing and overcoating migration imaging members XEROX CORPORTION (US) 1997-06-03 US disclosed
US-5534374-A Migration imaging members XEROX CORPORATION (US) 1996-07-09 US disclosed
EP-0673781-A1 Recording sheets containing amine salts and quaternary choline halides XEROX CORPORATION (US) 1995-09-27 EP disclosed
US-4565826-A HYPOTENSIVE, CARDIONASCULAR, ANTIULCER, ANTISECRETORY, GASTROINTESTINAL DISORDERS WILLIAM H. RORER, INC. (US) 1986-01-21 US disclosed
US-4564640-A Amidinoureas substituted in both the urea and amidino nitrogen positions WILLIAM H. RORER, INC. (US) 1986-01-14 US disclosed
EP-0078839-A4 HETEROCYCLIC AMIDINOUREAS. RORER INTERNAT OVERSEAS INC (US) 1984-07-25 EP disclosed
US-4436911-A HYPOTENSIVE, ANTISPASMODIC, ANTIULCER, ANTIPARASITIC WILLIAM H. RORER, INC. (US) 1984-03-13 US disclosed
EP-0078839-A1 HETEROCYCLIC AMIDINOUREAS RORER INTERNATIONAL (OVERSEAS) INC. (US) 1983-05-18 EP disclosed
WO-1982004047-A1 HETEROCYCLIC AMIDINOUREAS RORER INT OVERSEAS (US) 1982-11-25 WO disclosed
US-4178387-A ADMINISTERING AMIDINOUREAS WILLIAM H. RORER, INC. (US) 1979-12-11 US disclosed
US-4147804-A ANTIARRHYTHMIA AGENTS WILLIAM H. RORER, INC. (US) 1979-04-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100222580-A1 Process For The Preparation Of Onium Alkylsulfates Having A Low Halide Content STS, MRPS35, ARSA KDM4E 733/4885BLM 4589/4885CYP2D6 2179/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.