SCHEMBL3047838

SCHEMBL3047838

CCCNCc1ccc2[nH]c(-c3cc(OC)c(OS(C)(=O)=O)c4c3C(=O)NC4)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 9/20 0.40
KDR P35968 9/20 0.40
HTR1A P08908 1/20 0.35
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR7 P34969 1/20 0.35
HTR2B P41595 1/20 0.35
HTR5A P47898 1/20 0.35
HTR6 P50406 1/20 0.35
NQO2 P16083 1/20 0.34
CDK1 P06493 1/20 0.34
PKM P14618 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PARP1 P09874 2/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3034396 0.99 AURKA (0.40) AURKAKDRHTR1AHTR1DHTR1B
SCHEMBL3049157 0.94 AURKA (0.41) AURKAKDRHTR1AHTR1DHTR1B
SCHEMBL3048287 0.93 AURKA (0.40) AURKAKDRNQO2CDK1PKM
Hydrochloric Acid SCHEMBL3039578 0.93 AURKA (0.41) AURKAKDRHTR1AHTR1DHTR1B
SCHEMBL5043713 0.91 KDR (0.39) AURKAKDRNQO2CDK1PKM
Hydrochloric Acid SCHEMBL3046786 0.91 KDR (0.38) AURKAKDRNQO2CDK1PKM
Hydrochloric Acid SCHEMBL3047929 0.91 AURKA (0.38) AURKAKDRNQO2CDK1PKM
SCHEMBL3054784 0.90 AURKA (0.42) AURKAKDRHTR1AHTR1DHTR1B
Hydrochloric Acid SCHEMBL3046527 0.90 AURKA (0.42) AURKAKDRNQO2CDK1PKM
Hydrochloric Acid SCHEMBL3042710 0.90 AURKA (0.36) AURKAKDRNQO2CDK1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745641-B2 Nitrogen-containing heterocyclic compound KYOWA HAKKO KIRIN CO., LTD. (JP) 2010-06-29 US claimed