SCHEMBL30480865

SCHEMBL30480865

COc1cc2c(cc1Br)CCCN2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 10/20 0.56
HTR2A P28223 9/20 0.56
HTR2B P41595 6/20 0.56
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
ATM Q13315 1/20 0.38
CYP19A1 P11511 3/20 0.38
TLR9 Q9NR96 1/20 0.38
TLR8 Q9NR97 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
GAA P10253 1/20 0.38
THRB P10828 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18122551 1.00 HTR2C (0.56) HTR2CHTR2AHTR2BALDH1A1MAPT
Hydrochloric Acid SCHEMBL9331130 0.94 HTR2C (0.53) HTR2CHTR2AHTR2BALDH1A1MAPT
SCHEMBL18115471 0.90 HTR2C (0.64) HTR2CHTR2AHTR2BALDH1A1MAPT
SCHEMBL9331292 0.89 HTR2C (0.54) HTR2CHTR2AHTR2BALDH1A1MAPT
Hydrochloric Acid SCHEMBL9331810 0.87 HTR2C (0.53) HTR2CHTR2AHTR2BALDH1A1MAPT
SCHEMBL10912768 0.86 MAPT (0.45) HTR2CHTR2AHTR2BALDH1A1MAPT
Hydrochloric Acid SCHEMBL7373928 0.84 MAPT (0.44) HTR2CHTR2AHTR2BALDH1A1MAPT
SCHEMBL30340758 0.81 MAPT (0.43) HTR2CHTR2AHTR2BALDH1A1MAPT
SCHEMBL5468971 0.81 MAPT (0.43) HTR2CHTR2AHTR2BALDH1A1MAPT
SCHEMBL25405400 0.80 HTR2C (0.47) HTR2CHTR2AHTR2BALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116368128-A Heterocyclic compounds as CBP/EP300 bromodomain inhibitors 奥瑞基尼肿瘤有限公司 2023-06-30 CN disclosed