SCHEMBL30487148

SCHEMBL30487148

C[C@H](C(=O)N[C@@H]1COc2ccccc2[C@H]1N1CCC1)c1ccc(F)cc1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 9/20 0.66
P2RX7 Q99572 2/20 0.38
HTR2B P41595 3/20 0.37
PGR P06401 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20183016 1.00 GRM7 (0.66) GRM7P2RX7HTR2BPGRMEN1
SCHEMBL21542195 1.00 GRM7 (0.66) GRM7P2RX7HTR2BPGRMEN1
SCHEMBL21542196 1.00 GRM7 (0.66) GRM7P2RX7HTR2BPGRMEN1
SCHEMBL21542290 0.98 GRM7 (0.66) GRM7P2RX7HTR2BPGRMEN1
SCHEMBL21542288 0.98 GRM7 (0.66) GRM7P2RX7HTR2BPGRMEN1
SCHEMBL20182781 0.98 GRM7 (0.66) GRM7P2RX7HTR2BPGRMEN1
SCHEMBL20182845 0.92 GRM7 (0.64) GRM7P2RX7
SCHEMBL29909581 0.92 GRM7 (0.64) GRM7P2RX7
SCHEMBL21542311 0.92 GRM7 (0.64) GRM7P2RX7
SCHEMBL21542309 0.92 GRM7 (0.64) GRM7P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3541812-B1 MGLUR7 AGONIST COMPOUNDS FOR TREATING MGLUR7- REGULATED DISEASES, DISORDERS, OR CONDITIONS TAKEDA PHARMACEUTICALS CO (JP) 2023-06-14 EP disclosed