SCHEMBL30488019

SCHEMBL30488019

Nc1cc(-c2ccc(O)cc2)nc(N)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 3/20 0.61
ADORA1 P30542 3/20 0.50
ADORA2A P29274 2/20 0.50
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
NTSR1 P30989 1/20 0.48
LTA4H P09960 1/20 0.48
MKNK1 Q9BUB5 1/20 0.48
MKNK2 Q9HBH9 1/20 0.48
USP7 Q93009 1/20 0.47
MAPT P10636 2/20 0.47
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
PIK3CG P48736 2/20 0.46
CYP1A2 P05177 2/20 0.46
LMNA P02545 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28603599 1.00 DYRK1A (0.61) DYRK1AADORA1ADORA2AMEN1KMT2A
SCHEMBL6640763 0.81 NPC1 (0.46) DYRK1AMEN1KMT2AUSP7MAPT
SCHEMBL7379292 0.80 KDM4E (0.62) DYRK1AADORA1ADORA2AMAPTALDH1A1
SCHEMBL5511069 0.80 KDM4E (0.64) DYRK1AADORA1ADORA2AMAPTALDH1A1
SCHEMBL12443814 0.80 ADORA2A (0.73) DYRK1AADORA1ADORA2AMEN1KMT2A
SCHEMBL11645510 0.79 ADORA2A (0.79) DYRK1AADORA1ADORA2AMEN1KMT2A
SCHEMBL14496829 0.78 DYRK1A (0.54) DYRK1AADORA1ADORA2AKMT2AMAPT
SCHEMBL15757848 0.77 AURKA (0.56) DYRK1AADORA1ADORA2AMEN1KMT2A
Hydrochloric Acid SCHEMBL5542860 0.77 DYRK1A (0.53) DYRK1AADORA1ADORA2AKMT2AMAPT
SCHEMBL1388722 0.76 DYRK1A (1.00) DYRK1AADORA1MAPTALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113061116-B Aminopyrimidine compound, preparation method, composition and application thereof 上海医药工业研究院 2023-07-25 CN disclosed