SCHEMBL30495495

SCHEMBL30495495

O=C(CCCCCCCc1nc2ccccc2c(=O)[nH]1)NO

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.64
PARP2 Q9UGN5 2/20 0.64
HDAC3 O15379 1/20 0.58
HDAC4 P56524 1/20 0.58
HDAC1 Q13547 1/20 0.58
HDAC7 Q8WUI4 1/20 0.58
HDAC2 Q92769 1/20 0.58
HDAC10 Q969S8 1/20 0.58
HDAC11 Q96DB2 1/20 0.58
HDAC8 Q9BY41 1/20 0.58
HDAC6 Q9UBN7 1/20 0.58
HDAC9 Q9UKV0 1/20 0.58
HDAC5 Q9UQL6 1/20 0.58
TP53 P04637 1/20 0.58
G6PD P11413 1/20 0.58
PDE10A Q9Y233 1/20 0.58
PARP3 Q9Y6F1 6/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
RECQL P46063 1/20 0.57
CYP2C9 P11712 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29040111 1.00 PARP1 (0.64) PARP1PARP2HDAC3HDAC4HDAC1
SCHEMBL30495504 0.99 PARP1 (0.65) PARP1PARP2HDAC3HDAC4HDAC1
SCHEMBL29040068 0.95 PARP1 (0.67) PARP1PARP2TP53G6PDPDE10A
SCHEMBL29040039 0.90 PARP1 (0.74) PARP1PARP2PARP3SMN1; SMN2RECQL
SCHEMBL721483 0.84 HDAC3 (0.70) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL718972 0.84 HDAC3 (0.70) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL29040046 0.84 PARP1 (0.62) PARP1PARP2TP53G6PDPDE10A
SCHEMBL29040009 0.84 PARP1 (0.62) PARP1PARP2TP53G6PDPDE10A
SCHEMBL29040127 0.83 HDAC1 (0.60) PARP1PARP2HDAC3HDAC4HDAC1
SCHEMBL30495476 0.83 HDAC1 (0.60) PARP1PARP2HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116496224-B 4-Quinazolinone hydroxamic acid derivative, pharmaceutical composition and application thereof 武汉思瓴生物科技有限公司 2024-11-01 CN disclosed
CN-116496224-A 4-quinazolinone hydroxamic acid derivative, pharmaceutical composition and application thereof 武汉思瓴生物科技有限公司 2023-07-28 CN disclosed