SCHEMBL30530554

SCHEMBL30530554

O=C1CCN(C(=O)c2cncc(-c3ccccc3)c2)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 8/20 0.57
BRD2 P25440 2/20 0.57
HTT P42858 1/20 0.50
STAT3 P40763 1/20 0.48
LMNA P02545 2/20 0.47
RAB9A P51151 1/20 0.47
CYP11B1 P15538 2/20 0.46
CYP11B2 P19099 2/20 0.46
ALDH1A1 P00352 2/20 0.46
USP2 O75604 1/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
AVPR2 P30518 2/20 0.44
OXTR P30559 2/20 0.44
AVPR1A P37288 2/20 0.44
POLB P06746 1/20 0.44
HSD17B10 Q99714 1/20 0.44
HPGD P15428 1/20 0.43
CRBN Q96SW2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27197574 1.00 BRD4 (0.57) BRD4BRD2HTTSTAT3LMNA
SCHEMBL29598514 0.84 STAT3 (0.68) BRD4BRD2HTTSTAT3LMNA
SCHEMBL27197578 0.84 STAT3 (0.68) BRD4BRD2HTTSTAT3LMNA
SCHEMBL842907 0.80 HPGD (0.64) BRD4HTTSTAT3LMNARAB9A
SCHEMBL29598193 0.80 POLB (0.70) BRD4BRD2STAT3LMNARAB9A
SCHEMBL27197579 0.80 POLB (0.70) BRD4BRD2STAT3LMNARAB9A
SCHEMBL24499949 0.76 POLB (0.57) BRD4BRD2CYP11B2POLB
SCHEMBL29597188 0.76 POLB (0.55) BRD4BRD2STAT3CYP11B1CYP11B2
SCHEMBL27197589 0.76 POLB (0.55) BRD4BRD2STAT3CYP11B1CYP11B2
SCHEMBL30530566 0.75 STAT3 (0.62) BRD4HTTSTAT3RAB9ACYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116724034-A 2, 3-dihydro-4H-benzo [ B ] [1,4] oxazin-4-yl (5- (phenyl) -pyridin-3-yl) methanone derivatives and similar compounds as CYP11A1 inhibitors for the treatment of prostate cancer 奥赖恩公司 2023-09-08 CN claimed
CN-116724034-A 2, 3-dihydro-4H-benzo [ B ] [1,4] oxazin-4-yl (5- (phenyl) -pyridin-3-yl) methanone derivatives and similar compounds as CYP11A1 inhibitors for the treatment of prostate cancer 奥赖恩公司 2023-09-08 CN disclosed