SCHEMBL305356

SCHEMBL305356

O=C(O)NCn1cnc2ccccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN3 Q9H6Z9 1/20 0.60
SMN1; SMN2 Q16637 2/20 0.59
LMNA P02545 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
KDM4E B2RXH2 1/20 0.57
NPC1 O15118 1/20 0.57
APAF1 O14727 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
CYP11B1 P15538 2/20 0.54
CYP11B2 P19099 2/20 0.54
TNF P01375 1/20 0.54
HTT P42858 2/20 0.51
ASAH1 Q13510 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
GGPS1 O95749 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4359831 0.86 HDAC1 (0.58) EGLN3SMN1; SMN2LMNAL3MBTL1KDM4E
SCHEMBL16446114 0.86 KDM4E (0.60) EGLN3SMN1; SMN2LMNAL3MBTL1KDM4E
SCHEMBL10454788 0.84 EGLN3 (0.66) EGLN3SMN1; SMN2LMNAL3MBTL1KDM4E
SCHEMBL2867039 0.82 EGLN3 (0.62) EGLN3SMN1; SMN2LMNAL3MBTL1KDM4E
SCHEMBL2841675 0.81 EGLN3 (0.61) EGLN3SMN1; SMN2LMNAL3MBTL1KDM4E
SCHEMBL1035783 0.78 EGLN3 (0.71) EGLN3SMN1; SMN2LMNAL3MBTL1KDM4E
Hydrogen Sulfide SCHEMBL28767930 0.77 EGLN3 (0.69) EGLN3SMN1; SMN2LMNAL3MBTL1KDM4E
Hydrochloric Acid SCHEMBL1082612 0.77 EGLN3 (0.69) EGLN3SMN1; SMN2LMNAL3MBTL1KDM4E
SCHEMBL8327961 0.76 TDP1 (0.63) EGLN3SMN1; SMN2LMNAKDM4ENPC1
SCHEMBL6006482 0.75 TDP1 (0.58) EGLN3SMN1; SMN2LMNAL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 60 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0513409-B1 Use of a microbicide agent for making concrete shingles RIEDEL DE HAEN AG (DE) 1996-07-24 EP claimed
US-12089593-B2 Compositions and methods for treating and preventing dust mite infestation DANSTAR FERMENT AG (CH) 2024-09-17 US disclosed
US-20190090482-A1 COMPOSITIONS AND METHODS FOR TREATING AND PREVENTING DUST MITE INFESTATION DANSTAR FERMENT AG (CH) 2019-03-28 US disclosed
EP-3432710-A1 COMPOSITIONS AND METHODS FOR TREATING AND PREVENTING DUST MITE INFESTATION Evolva SA (CH) 2019-01-30 EP disclosed
WO-2017162877-A1 COMPOSITIONS AND METHODS FOR TREATING AND PREVENTING DUST MITE INFESTATION EVOLVA SA (CH) 2017-09-28 WO disclosed
EP-2323485-B1 ANTI-ALLERGEN COMBINATIONS OF CALCIUM AND LANTHANUM SALTS JANSSEN PHARMACEUTICA NV (BE) 2013-10-16 EP disclosed
CN-101658183-B Mildew removing and preventing agent for interior walls of building DU ZHIGANG 2013-07-31 CN disclosed
CN-101535464-B Premoistened cleaning disposable substrate CIBA HOLDING INC 2012-01-18 CN disclosed
US-8093199-B2 Premoistened cleaning disposable substrate and method of incorporation of a cleaning composition into said substrate BASF SE (DE) 2012-01-10 US disclosed
EP-2082021-B1 PREMOISTENED CLEANING DISPOSABLE SUBSTRATE BASF SE (DE) 2011-08-03 EP disclosed
EP-0469357-A1 1-[pyri(mi)dyl-(2)]-5-hydroxypyrazole microbicides BAYER AG (DE) 1992-02-05 EP disclosed
US-4966974-A IN PLANT PROTECTION; IMPROVED STABILITY TO HYDROLYSIS BAYER AKTIENGESELLSCHAFT (DE) 1990-10-30 US disclosed
EP-0195238-B1 N-SULPHENYLIZED INDAZOLES CONTAINING FLUORINE, PROCESS FOR THEIR PREPARATION AND THEIR USE BAYER AG (DE) 1989-03-29 EP disclosed
EP-0142785-B1 TRIHALO-ALLYLTHIOCYANATES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN MICROBICIDAL AGENTS BAYER AG (DE) 1987-03-18 EP disclosed
EP-0148442-B1 HALOGENATED SULFIDES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN MICROBICIDAL COMPOSITIONS BAYER AG (DE) 1987-01-21 EP disclosed
EP-0121054-B1 N-SULPHENYLIZED HYDANTOINS, PROCESS FOR THEIR PREPARATION AND THEIR MICROBICIDAL USE BAYER AG (DE) 1986-12-03 EP disclosed
EP-0148442-A2 Halogenated sulfides, process for their preparation and their use in microbicidal compositions BAYER AG (DE) 1985-07-17 EP disclosed
EP-0142785-A2 Trihalo-allylthiocyanates, process for their preparation and their use in microbicidal agents BAYER AG (DE) 1985-05-29 EP disclosed
US-4395274-A BENZIMIDAZOLYL-ALKYL-CARBONATES AND A CHLORINATED PHENOLIC COMPOUND BAYER AKTIENGESELLSCHAFT (DE) 1983-07-26 US disclosed
US-4026934-A INSECTICIDES, ACARICIDES, FUNGICIDES BAYER AKTIENGESELLSCHAFT (DT) 1977-05-31 US disclosed