SCHEMBL30539133

SCHEMBL30539133

C=CC(=O)Nc1cc(Nc2nccc(-c3cn(C)c4cc(OC)ccc34)n2)c(OC)cc1N(C)CCNC

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.85
IGF1R P08069 1/20 0.85
MLNR O43193 1/20 0.73
KDM1A O60341 1/20 0.73
ABCB11 O95342 1/20 0.73
ERBB2 P04626 1/20 0.73
INSR P06213 1/20 0.73
CHRM2 P08172 1/20 0.73
HTR1A P08908 1/20 0.73
ADORA3 P0DMS8 1/20 0.73
DRD2 P14416 1/20 0.73
NQO2 P16083 1/20 0.73
ADRA2C P18825 1/20 0.73
DRD1 P21728 1/20 0.73
ERBB3 P21860 1/20 0.73
SLC6A2 P23975 1/20 0.73
HTR2A P28223 1/20 0.73
HTR2C P28335 1/20 0.73
ADORA2A P29274 1/20 0.73
SLC6A4 P31645 1/20 0.73

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17683157 1.00 EGFR (0.85) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL17683059 0.93 EGFR (0.86) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL29860673 0.92 EGFR (1.00) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL14661086 0.92 EGFR (1.00) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL30379658 0.92 EGFR (1.00) EGFRIGF1RMLNRKDM1AABCB11
Hydrochloric Acid SCHEMBL30735856 0.91 EGFR (0.99) EGFRIGF1RMLNRKDM1AABCB11
Hydrochloric Acid SCHEMBL26637892 0.91 EGFR (0.99) EGFRIGF1RMLNRKDM1AABCB11
Hydrochloric Acid SCHEMBL30735819 0.91 EGFR (0.99) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL30682157 0.89 EGFR (0.95) EGFRIGF1RMLNRKDM1AABCB11
SCHEMBL22509231 0.89 EGFR (0.87) EGFRIGF1RMLNRKDM1AABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402143-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2024-01-16 CN disclosed
CN-111187221-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-26 CN disclosed
CN-111171000-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-01 CN disclosed