SCHEMBL30580392

SCHEMBL30580392

COc1cc(NC(=O)c2cscn2)ccc1-c1cnc2[nH]ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 4/20 0.53
TNIK Q9UKE5 2/20 0.51
BRD4 O60885 1/20 0.46
POLQ O75417 1/20 0.45
CDK8 P49336 7/20 0.45
IMPDH2 P12268 1/20 0.44
ROCK2 O75116 2/20 0.44
KDM4E B2RXH2 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PIK3C3 Q8NEB9 1/20 0.42
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42
PLK4 O00444 1/20 0.42
DCLK1 O15075 1/20 0.42
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
PAK4 O96013 1/20 0.42
CHEK2 O96017 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29072630 1.00 GRM4 (0.53) GRM4TNIKBRD4POLQCDK8
SCHEMBL30580382 0.86 SMN1; SMN2 (0.60) GRM4TNIKBRD4CDK8KDM4E
SCHEMBL29072544 0.86 SMN1; SMN2 (0.60) GRM4TNIKBRD4CDK8KDM4E
SCHEMBL30580401 0.83 TNIK (0.57) TNIKBRD4CDK8IMPDH2ROCK2
SCHEMBL29072546 0.83 TNIK (0.57) TNIKBRD4CDK8IMPDH2ROCK2
SCHEMBL30580375 0.82 PIK3C3 (0.55) TNIKBRD4POLQCDK8IMPDH2
SCHEMBL29072979 0.82 PIK3C3 (0.55) TNIKBRD4POLQCDK8IMPDH2
SCHEMBL30580376 0.82 TNIK (0.54) TNIKBRD4POLQCDK8IMPDH2
SCHEMBL29072559 0.82 TNIK (0.54) TNIKBRD4POLQCDK8IMPDH2
SCHEMBL29072554 0.82 TNIK (0.54) TNIKBRD4POLQCDK8IMPDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116768886-A N- (4- (1H-pyrrolo [2,3-b ] pyridin-5-yl) phenyl) amide derivatives, preparation and use thereof 安徽医科大学 2023-09-19 CN disclosed