SCHEMBL30587265

SCHEMBL30587265

N#Cc1c(N)sc2ccc(F)c(-c3c4c(c5c(N6C7CCC6CNC7)ncnc5c3F)COC4)c12

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KRAS P01116 2/20 0.40
RPS6KB1 P23443 1/20 0.31
AKT1 P31749 1/20 0.31
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26113820 1.00 KRAS (0.40) KRASRPS6KB1AKT1LRRK2
SCHEMBL30776336 0.95 KRAS (0.39) KRASRPS6KB1AKT1
SCHEMBL26542738 0.95 KRAS (0.39) KRASRPS6KB1AKT1
SCHEMBL30776522 0.87 KRAS (0.38) KRAS
SCHEMBL26546016 0.87 KRAS (0.38) KRAS
SCHEMBL30776400 0.86 KRAS (0.34) KRASRPS6KB1AKT1LRRK2
SCHEMBL26542838 0.86 KRAS (0.34) KRASRPS6KB1AKT1LRRK2
SCHEMBL26544287 0.86 KRAS (0.40) KRASRPS6KB1AKT1
SCHEMBL26542503 0.86 KRAS (0.38) KRAS
SCHEMBL30776294 0.85 KRAS (0.37) KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250289830-A1 KRAS INHIBITORS ELI LILLY AND COMPANY 2025-09-18 US disclosed
US-12351591-B2 KRas inhibitors ELI LILLY AND COMPANY (US) 2025-07-08 US disclosed
EP-4499233-A1 KRAS INHIBITORS Eli Lilly and Company (US) 2025-02-05 EP disclosed
CN-119095853-A KRAS inhibitors 伊莱利利公司 2024-12-06 CN disclosed
US-20240043451-A1 KRAS INHIBITORS ELI LILLY AND COMPANY 2024-02-08 US disclosed
WO-2023183585-A1 KRAS INHIBITORS ELI LILLY AND COMPANY (US) 2023-09-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240043451-A1 KRAS INHIBITORS KRAS, NRAS, HRAS KRAS 1/4885RPS6KB1 764/4885AKT1 40/4885
US-12351591-B2 KRas inhibitors KRAS, NRAS, HRAS KRAS 1/4885RPS6KB1 764/4885AKT1 40/4885
US-20250289830-A1 KRAS INHIBITORS KRAS, NRAS, HRAS KRAS 1/4885RPS6KB1 764/4885AKT1 40/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.