SCHEMBL30604173

SCHEMBL30604173

c1cncc(-c2ccc3ncccc3c2)c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.75
RAB9A P51151 2/20 0.75
POLB P06746 1/20 0.75
CYP2A6 P11509 3/20 0.70
CYP11B1 P15538 6/20 0.66
CYP11B2 P19099 6/20 0.66
CYP19A1 P11511 4/20 0.66
CYP17A1 P05093 3/20 0.66
DYRK1A Q13627 1/20 0.60
QPCT Q16769 1/20 0.55
QPCTL Q9NXS2 1/20 0.55
KDM4E B2RXH2 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
PIK3CA P42336 2/20 0.55
ALDH1A1 P00352 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
PIK3CD O00329 1/20 0.53
PIP5K1C O60331 1/20 0.53
PI4KA P42356 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21264426 1.00 NPC1 (0.75) NPC1RAB9APOLBCYP2A6CYP11B1
SCHEMBL23543013 0.87 CYP2A6 (0.58) NPC1RAB9APOLBCYP2A6CYP11B1
SCHEMBL30743 0.87 NPC1 (1.00) NPC1RAB9APOLBCYP2A6DYRK1A
SCHEMBL29757180 0.87 NPC1 (1.00) NPC1RAB9APOLBCYP2A6DYRK1A
SCHEMBL23543024 0.86 CYP2A6 (0.61) NPC1RAB9APOLBCYP2A6CYP11B1
SCHEMBL19297863 0.86 NPC1 (0.75) NPC1RAB9APOLBCYP2A6CYP11B1
SCHEMBL23467163 0.86 CYP11B1 (0.66) NPC1RAB9APOLBCYP2A6CYP11B1
SCHEMBL443618 0.83 NPC1 (0.84) NPC1RAB9APOLBCYP2A6CYP11B1
SCHEMBL30592751 0.83 NPC1 (0.84) NPC1RAB9APOLBCYP2A6CYP11B1
SCHEMBL12075055 0.83 NPC1 (0.84) NPC1RAB9APOLBCYP2A6CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116745291-A N- (2- (4-cyanothiazolidin-3-yl) -2-oxoethyl) -quinoline-4-carboxamide 阿斯利康(瑞典)有限公司 2023-09-12 CN disclosed