SCHEMBL30627720

SCHEMBL30627720

Cc1nsc(-c2nnc3n2CCN(C(=O)C2CC2)[C@@H]3C)n1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 20/20 0.67
KCNH2 Q12809 10/20 0.67
CYP2C9 P11712 3/20 0.67
CYP2C19 P33261 3/20 0.67
CYP1A2 P05177 2/20 0.67
CYP3A4 P08684 2/20 0.67
TACR1 P25103 3/20 0.66
CYP2D6 P10635 1/20 0.66
TACR2 P21452 4/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30627839 0.94 TACR3 (0.63) TACR3KCNH2CYP2C9CYP2C19CYP1A2
SCHEMBL29967223 0.87 TACR3 (0.74) TACR3KCNH2CYP2C9CYP2C19CYP1A2
SCHEMBL30627779 0.83 TACR3 (0.50) TACR3KCNH2CYP2C9CYP2C19CYP1A2
SCHEMBL30627826 0.82 TACR3 (0.64) TACR3KCNH2CYP2C9CYP2C19CYP1A2
SCHEMBL30627726 0.81 TACR3 (0.81) TACR3KCNH2CYP2C9CYP2C19CYP1A2
SCHEMBL29941569 0.81 TACR3 (0.68) TACR3KCNH2CYP2C9CYP2C19CYP1A2
SCHEMBL17005283 0.80 TACR3 (1.00) TACR3KCNH2CYP2C9CYP2C19CYP1A2
SCHEMBL16143075 0.80 TACR3 (1.00) TACR3KCNH2CYP2C9CYP2C19CYP1A2
SCHEMBL16143073 0.80 TACR3 (1.00) TACR3KCNH2CYP2C9CYP2C19CYP1A2
SCHEMBL26963887 0.80 TACR3 (0.44) TACR3KCNH2CYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112272670-B Di-ring derivative-containing inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-12 CN disclosed