SCHEMBL30644271

SCHEMBL30644271

Brc1ccc(N2CCN3CCOC[C@H]3C2)nc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.51
SOS1 Q07889 11/20 0.42
LRRK2 Q5S007 5/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
MAP4K4 O95819 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5623842 0.86 GRIN2D (0.48) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL1781248 0.85 MAP4K4 (0.53) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL20491766 0.85 AKR1C3 (0.52) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL20456794 0.85 AKR1C3 (0.52) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL20456700 0.85 AKR1C3 (0.52) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL21812428 0.85 AKR1C3 (0.53) AKR1C3GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL23253058 0.84 SOS1 (0.46) SOS1LRRK2
SCHEMBL20456847 0.84 SOS1 (0.42) SOS1LRRK2MAP4K4
SCHEMBL20456845 0.84 SOS1 (0.42) SOS1LRRK2MAP4K4
SCHEMBL20469097 0.84 SOS1 (0.46) SOS1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117003755-A Pyrazolopyridazinone derivatives, compositions and uses thereof 北京伯汇生物技术有限公司 2023-11-07 CN disclosed