SCHEMBL30646121

SCHEMBL30646121

CCC1(C)CCc2nc(Cl)ccc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.39
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31
GRIN2C Q14957 1/20 0.31
GRIN3A Q8TCU5 1/20 0.31
TDP2 O95551 1/20 0.30
NSD2 O96028 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30646092 0.85 GRM5 (0.36) GRM5TDP2NSD2
SCHEMBL30646147 0.84 GRM5 (0.36) GRM5ESR1ESR2GRIN2DGRIN3B
SCHEMBL30646090 0.82 GRM5 (0.45) GRM5ESR1ESR2
SCHEMBL4683297 0.81 GRM5 (0.55) GRM5TDP2NSD2
SCHEMBL30646083 0.81 GRM5 (0.55) GRM5TDP2NSD2
SCHEMBL16801069 0.77 CYP19A1 (0.36) GRM5ESR1ESR2GRIN2DGRIN3B
SCHEMBL30646085 0.77 GRM5 (0.39) GRM5TDP2NSD2
SCHEMBL31668731 0.76 GRM5 (0.37) GRM5TDP2NSD2
SCHEMBL4433359 0.76 GRM5 (0.34) GRM5
SCHEMBL13669670 0.76 MEN1 (0.34) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4543437-A1 3-?HSD1 INHIBITORS AND COMPOSITIONS AND USES THEREOF THE CLEVELAND CLINIC FOUNDATION (US) 2025-04-30 EP disclosed
WO-2023250480-A1 3-βHSD1 INHIBITORS AND COMPOSITIONS AND USES THEREOF THE CLEVELAND CLINIC FOUNDATION (US) 2023-12-28 WO disclosed