SCHEMBL30663261

SCHEMBL30663261

CCc1cc2ccc(CN3CCN(c4ccccn4)CC3)cc2[nH]c1=O

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 19/20 0.75
PARP2 Q9UGN5 9/20 0.64
KCNH2 Q12809 4/20 0.64
ALDH1A1 P00352 1/20 0.54
TNK1 Q13470 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8067001 1.00 PARP1 (0.75) PARP1PARP2KCNH2ALDH1A1TNK1
SCHEMBL8078172 0.89 PARP1 (0.62) PARP1PARP2KCNH2ALDH1A1TNK1
SCHEMBL8067063 0.89 PARP1 (0.67) PARP1PARP2KCNH2
SCHEMBL8076822 0.87 PARP1 (0.68) PARP1PARP2KCNH2TNK1
SCHEMBL25092969 0.86 PARP1 (1.00) PARP1PARP2
SCHEMBL30893587 0.86 PARP1 (1.00) PARP1PARP2
SCHEMBL8071284 0.84 PARP1 (0.71) PARP1PARP2KCNH2
SCHEMBL8070707 0.82 PARP1 (0.69) PARP1PARP2KCNH2
SCHEMBL8075135 0.82 PARP1 (1.00) PARP1PARP2KCNH2TNK1
SCHEMBL8076591 0.82 PARP1 (0.71) PARP1PARP2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117177972-A PARP1 inhibitors and uses thereof 新特拉有限公司 2023-12-05 CN disclosed