SCHEMBL30690342

SCHEMBL30690342

Cc1cc([C@@H](C)N)c2nc(-c3c(F)cccc3F)n(C)c(=O)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 1/20 0.35
AKT2 P31751 1/20 0.35
AKT3 Q9Y243 1/20 0.35
PIK3CB P42338 1/20 0.35
GPR139 Q6DWJ6 1/20 0.33
ADRA1A P35348 1/20 0.33
KCNH2 Q12809 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
DHODH Q02127 3/20 0.33
WEE1 P30291 1/20 0.31
PTGES O14684 3/20 0.31
TRPV4 Q9HBA0 1/20 0.31
AADAT Q8N5Z0 1/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31
PDE4D Q08499 1/20 0.31
PDE7A Q13946 1/20 0.31
PDE7B Q9NP56 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29139165 1.00 AKT1 (0.35) AKT1AKT2AKT3PIK3CBGPR139
SCHEMBL29139168 1.00 AKT1 (0.35) AKT1AKT2AKT3PIK3CBGPR139
SCHEMBL25361230 0.87 AKT1 (0.37) AKT1AKT2AKT3DHODH
SCHEMBL30495135 0.87 AKT1 (0.37) AKT1AKT2AKT3DHODH
SCHEMBL25361232 0.87 AKT1 (0.37) AKT1AKT2AKT3DHODH
SCHEMBL25360386 0.84 ADORA2A (0.39) AKT1AKT2AKT3
SCHEMBL25360382 0.84 ADORA2A (0.39) AKT1AKT2AKT3
SCHEMBL30495001 0.84 ADORA2A (0.39) AKT1AKT2AKT3
SCHEMBL25361392 0.82 POLB (0.35) AKT1AKT2AKT3ADRA1AKCNH2
SCHEMBL25361398 0.82 POLB (0.35) AKT1AKT2AKT3ADRA1AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117362281-A PI3K inhibitor and preparation method and application thereof 海创药业股份有限公司 2024-01-09 CN disclosed