SCHEMBL30693201

SCHEMBL30693201

CC(C)(C)OC(=O)N1CC[C@@H](N2CCN(Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)C2=O)[C@H](c2ccc(Cl)c(Cl)c2)C1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.47
TP53 P04637 1/20 0.43
TACR2 P21452 7/20 0.42
TAC3 Q9UHF0 1/20 0.42
TACR3 P29371 3/20 0.41
STS P08842 1/20 0.39
MC4R P32245 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1971060 1.00 TACR1 (0.47) TACR1TP53TACR2TAC3TACR3
SCHEMBL15397629 0.88 TACR1 (0.43) TACR1TACR2TAC3TACR3
SCHEMBL1968714 0.85 TACR1 (0.60) TACR1TACR2TAC3TACR3
SCHEMBL1971144 0.77 USP30 (0.51) TACR1TP53TACR2TAC3TACR3
Hydrochloric Acid SCHEMBL1969632 0.77 TACR1 (0.38) TACR1TACR2TAC3TACR3
SCHEMBL1970339 0.77 TACR1 (0.53) TACR1TACR2TAC3TACR3
SCHEMBL30693211 0.77 TACR1 (0.53) TACR1TACR2TAC3TACR3
SCHEMBL4150434 0.77 TACR1 (0.49) TACR1TACR2TAC3TACR3STS
SCHEMBL13801311 0.77 TACR1 (0.49) TACR1TACR2TAC3TACR3STS
SCHEMBL13801316 0.77 TACR1 (0.49) TACR1TACR2TAC3TACR3STS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE49686-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2023-10-10 US disclosed