SCHEMBL30701799

SCHEMBL30701799

COc1ccc(CNc2ccc(N3CCOCC3)c(C(=O)NCC(C)(C)C)c2)cc1F

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH2 P05091 1/20 0.78
GAA P10253 11/20 0.60
KDM4E B2RXH2 7/20 0.60
HSD17B10 Q99714 5/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
HDAC3 O15379 3/20 0.55
HDAC1 Q13547 3/20 0.55
HDAC2 Q92769 3/20 0.55
HDAC8 Q9BY41 3/20 0.55
HDAC6 Q9UBN7 3/20 0.55
ALDH1A1 P00352 6/20 0.53
ALOX15 P16050 3/20 0.53
MAPK1 P28482 2/20 0.53
MAPT P10636 1/20 0.53
TUBB4A P04350 1/20 0.52
TUBB P07437 1/20 0.52
TUBA3C P0DPH7 1/20 0.52
TUBA1B P68363 1/20 0.52
TUBA4A P68366 1/20 0.52
TUBB4B P68371 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29106413 1.00 ALDH2 (0.78) ALDH2GAAKDM4EHSD17B10SMN1; SMN2
SCHEMBL29106286 0.95 ALDH2 (0.78) ALDH2GAAKDM4EHSD17B10SMN1; SMN2
SCHEMBL30701807 0.95 ALDH2 (0.78) ALDH2GAAKDM4EHSD17B10SMN1; SMN2
SCHEMBL29106300 0.94 ALDH2 (0.77) ALDH2GAAKDM4EHSD17B10SMN1; SMN2
SCHEMBL29106341 0.92 ALDH2 (0.73) ALDH2GAAKDM4EHSD17B10SMN1; SMN2
SCHEMBL29106345 0.91 ALDH2 (0.81) ALDH2GAAKDM4EHSD17B10SMN1; SMN2
SCHEMBL30701810 0.89 ALDH2 (0.78) ALDH2GAAKDM4EHSD17B10SMN1; SMN2
SCHEMBL29106415 0.89 ALDH2 (0.78) ALDH2GAAKDM4EHSD17B10SMN1; SMN2
SCHEMBL30701802 0.89 ALDH2 (0.75) ALDH2GAAKDM4EHSD17B10SMN1; SMN2
SCHEMBL29106378 0.89 ALDH2 (0.75) ALDH2GAAKDM4EHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109942537-B ALDH2 agonist, preparation method and application thereof 中国人民解放军第二军医大学 2023-11-17 CN claimed