SCHEMBL30703117

SCHEMBL30703117

C[Si](C)(C)CCOCn1c(-c2ccc(CN3CCC(F)(F)CC3)cc2)cc2c(Cl)ncnc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.36
TLR7 Q9NYK1 2/20 0.36
MAP3K11 Q16584 1/20 0.34
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
KCNH2 Q12809 1/20 0.32
BRD4 O60885 1/20 0.32
PDE1B Q01064 4/20 0.31
WNT1 P04628 1/20 0.31
CLK2 P49760 1/20 0.31
CLK3 P49761 1/20 0.31
DYRK1A Q13627 1/20 0.31
CYP2D6 P10635 1/20 0.31
CASP6 P55212 1/20 0.31
SSTR5 P35346 1/20 0.31
GRM2 Q14416 1/20 0.31
HSP90AA1 P07900 1/20 0.30
CNR1 P21554 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21484352 1.00 HRH3 (0.36) HRH3TLR7MAP3K11JAK2JAK1
SCHEMBL21484313 0.86 MEN1 (0.38) JAK2JAK1TYK2JAK3KCNH2
SCHEMBL30862663 0.83 NPC1 (0.35) PDE1B
SCHEMBL21484354 0.83 TLR7 (0.34) HRH3TLR7JAK2JAK1TYK2
SCHEMBL24541937 0.80 NPC1 (0.36)
SCHEMBL21409297 0.80 NPC1 (0.36)
SCHEMBL30862665 0.79 TDP1 (0.38) PDE1B
SCHEMBL17290075 0.78 CYP11B1 (0.39)
SCHEMBL17289652 0.78 MCHR1 (0.43) HRH3KCNH2
SCHEMBL21484350 0.78 PIM1 (0.40) HRH3KCNH2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112812117-B Novel crystal form of BTK inhibitor and preparation method thereof 中国医药研究开发中心有限公司 2023-12-22 CN disclosed