SCHEMBL30715263

SCHEMBL30715263

COC(=O)[C@@H]1CCc2nc(Cl)cc(=O)n21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.41
KMT2A Q03164 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
MEN1 O00255 2/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35
F11 P03951 2/20 0.35
TDP1 Q9NUW8 1/20 0.34
CHRNB4 P30926 2/20 0.34
CHRNA3 P32297 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PREP P48147 1/20 0.33
CASP1 P29466 1/20 0.33
CASP3 P42574 1/20 0.33
CASP8 Q14790 1/20 0.33
OPRM1 P35372 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16754160 0.85 TSHR (0.38) LMNAKMT2ASMN1; SMN2MEN1TDP1
SCHEMBL19470053 0.82 ACE (0.37) LMNAF11TDP1PREPCASP1
SCHEMBL29143359 0.82 ACE (0.37) LMNAF11TDP1PREPCASP1
SCHEMBL10189678 0.76 ADRB3 (0.41) KMT2ASMN1; SMN2MEN1ALDH1A1OPRM1
SCHEMBL11964111 0.76 ADRB3 (0.41) KMT2ASMN1; SMN2MEN1ALDH1A1OPRM1
SCHEMBL19595725 0.72 GAA (0.38) KMT2AMEN1ALDH1A1CYP3A4
SCHEMBL15079202 0.72 GAA (0.38) KMT2AMEN1ALDH1A1CYP3A4
SCHEMBL27070540 0.71 CYP1A2 (0.40) KMT2ACYP2C19
SCHEMBL19584519 0.70 KMT2A (0.35) LMNAKMT2AMEN1CASP3
SCHEMBL19618711 0.70 KDM4E (0.40) KMT2ASMN1; SMN2MEN1F11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402117-B Preparation method of 4-pyrimidinone derivative 南京威凯尔生物医药科技有限公司 2024-03-19 CN disclosed
CN-117402117-A Preparation method of 4-pyrimidinone derivative 南京威凯尔生物医药科技有限公司 2024-01-16 CN disclosed