SCHEMBL30718355

SCHEMBL30718355

CC1(C)c2nc(-c3cc(Cl)cc(Cl)c3)c(Nc3ccc(F)cc3)n2CCN1C(=O)CN

nearest known ligand 0.85

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 13/20 0.85
CYP3A4 P08684 1/20 0.83
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
TACR3 P29371 1/20 0.35
CYP2C19 P33261 1/20 0.35
DPP4 P27487 2/20 0.32
DPP8 Q6V1X1 2/20 0.32
DPP9 Q86TI2 2/20 0.32
DPP7 Q9UHL4 2/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
CNR1 P21554 1/20 0.32
DGAT2 Q96PD7 1/20 0.32
PIK3CD O00329 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30718361 0.96 KCNH2 (0.82) KCNH2CYP3A4CYP1A2CYP2C9TACR3
SCHEMBL30718427 0.92 KCNH2 (0.81) KCNH2CYP3A4
SCHEMBL1049907 0.92 KCNH2 (1.00) KCNH2CYP3A4CYP1A2CYP2C9TACR3
SCHEMBL30718360 0.92 KCNH2 (1.00) KCNH2CYP3A4CYP1A2CYP2C9TACR3
SCHEMBL30718406 0.92 KCNH2 (0.87) KCNH2CYP3A4CYP1A2CYP2C9TACR3
Ganaplacide SCHEMBL1047381 0.91 KCNH2 (1.00) KCNH2CYP3A4CYP1A2CYP2C9TACR3
SCHEMBL30718420 0.91 KCNH2 (0.84) KCNH2CYP3A4PIK3CD
SCHEMBL30718378 0.90 KCNH2 (0.84) KCNH2CYP3A4CYP1A2CYP2C9TACR3
SCHEMBL30718433 0.90 KCNH2 (0.77) KCNH2CYP3A4CYP1A2CYP2C9TACR3
SCHEMBL30718447 0.90 KCNH2 (0.83) KCNH2CYP3A4CYP1A2CYP2C9TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024006970-A2 ANTIMALARIAL COMPOUNDS THE SCRIPPS RESEARCH INSTITUTE (US) 2024-01-04 WO claimed
WO-2024006971-A2 ANTIMALARIAL COMPOUNDS THE SCRIPPS RESEARCH INSTITUTE (US) 2024-01-04 WO claimed
WO-2024006970-A2 ANTIMALARIAL COMPOUNDS THE SCRIPPS RESEARCH INSTITUTE (US) 2024-01-04 WO disclosed
WO-2024006971-A2 ANTIMALARIAL COMPOUNDS THE SCRIPPS RESEARCH INSTITUTE (US) 2024-01-04 WO disclosed