SCHEMBL30719113

SCHEMBL30719113

CCOC(=O)c1cc(C(=O)OCC)n(CC(=O)c2cccc(C#N)c2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.48
GSK3B P49841 1/20 0.44
GRM5 P41594 1/20 0.43
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
GAA P10253 2/20 0.40
ALDH1A1 P00352 2/20 0.40
RXFP1 Q9HBX9 1/20 0.40
PDCD1 Q15116 1/20 0.39
CD274 Q9NZQ7 1/20 0.39
CYP1A2 P05177 1/20 0.39
FNTA P49354 1/20 0.39
FNTB P49356 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 2/20 0.39
HRH2 P25021 1/20 0.39
HRH1 P35367 1/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21630625 1.00 ELANE (0.48) ELANEGSK3BGRM5KMT2AMEN1
SCHEMBL14725968 0.85 ELANE (0.50) ELANEKMT2AALDH1A1SMN1; SMN2POLB
SCHEMBL28560572 0.80 SMN1; SMN2 (0.46) KMT2AMEN1GAAALDH1A1CYP1A2
SCHEMBL29977154 0.80 SMN1; SMN2 (0.46) KMT2AMEN1GAAALDH1A1CYP1A2
SCHEMBL28554740 0.79 KMT2A (0.48) KMT2AMEN1GAAALDH1A1CYP1A2
SCHEMBL28546956 0.79 SMN1; SMN2 (0.40) KMT2AMEN1GAACYP1A2SMN1; SMN2
SCHEMBL23112463 0.78 NOTUM (0.49) KMT2AMEN1GAAALDH1A1CYP1A2
SCHEMBL29977559 0.78 NOTUM (0.49) KMT2AMEN1GAAALDH1A1CYP1A2
SCHEMBL29977403 0.77 SMN1; SMN2 (0.43) ELANEKMT2AMEN1GAAALDH1A1
SCHEMBL28556855 0.77 SMN1; SMN2 (0.43) ELANEKMT2AMEN1GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113166153-B Fused pyrazine derivatives as A2A/A2B inhibitors 因赛特公司 2024-11-01 CN disclosed
CN-117304191-A Fused pyrazine derivatives as A2A/A2B inhibitors 因赛特公司 2023-12-29 CN disclosed