Onfasprodil

Onfasprodil

SCHEMBL30727985

Oc1ccc([C@@H](O)CN2C[C@H]3C[C@H](Oc4ccccc4F)C[C@H]3C2)nc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 20/20 1.00
GRIN2B Q13224 20/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Onfasprodil SCHEMBL30648114 1.00 GRIN1 (1.00) GRIN1GRIN2B
Onfasprodil SCHEMBL17633369 1.00 GRIN1 (1.00) GRIN1GRIN2B
Onfasprodil SCHEMBL29346467 1.00 GRIN1 (1.00) GRIN1GRIN2B
Onfasprodil SCHEMBL29882782 1.00 GRIN1 (1.00) GRIN1GRIN2B
Onfasprodil SCHEMBL20086359 1.00 GRIN1 (1.00) GRIN1GRIN2B
Onfasprodil SCHEMBL17633403 1.00 GRIN1 (1.00) GRIN1GRIN2B
Onfasprodil SCHEMBL17633258 1.00 GRIN1 (1.00) GRIN1GRIN2B
Onfasprodil SCHEMBL30648127 1.00 GRIN1 (1.00) GRIN1GRIN2B
Onfasprodil SCHEMBL17633362 1.00 GRIN1 (1.00) GRIN1GRIN2B
Onfasprodil SCHEMBL20983421 1.00 GRIN1 (1.00) GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025264860-A2 METHODS OF TREATING POST-COVID AIRWAY DISEASE YALE UNIVERSITY (US) 2025-12-26 WO claimed
EP-4629989-A2 TREATMENT OR PREVENTION OF DEPRESSIVE DISORDERS THROUGH COMBINATION THERAPY Freedom Biosciences, Inc. (US) 2025-10-15 EP claimed
WO-2025120013-A1 COMPOSITIONS AND METHODS FOR TREATING DEPRESSION DISORDERS NOVARTIS AG (CH) 2025-06-12 WO claimed
WO-2024123935-A2 TREATMENT OR PREVENTION OF DEPRESSIVE DISORDERS THROUGH COMBINATION THERAPY FREEDOM BIOSCIENCES, INC. (US) 2024-06-13 WO claimed
WO-2025264860-A2 METHODS OF TREATING POST-COVID AIRWAY DISEASE YALE UNIVERSITY (US) 2025-12-26 WO disclosed
EP-4649143-A1 ENGINEERED KETOREDUCTASE POLYPEPTIDES Novartis AG (CH) 2025-11-19 EP disclosed
EP-4629989-A2 TREATMENT OR PREVENTION OF DEPRESSIVE DISORDERS THROUGH COMBINATION THERAPY Freedom Biosciences, Inc. (US) 2025-10-15 EP disclosed
WO-2025120013-A1 COMPOSITIONS AND METHODS FOR TREATING DEPRESSION DISORDERS NOVARTIS AG (CH) 2025-06-12 WO disclosed
WO-2025120013-A1 COMPOSITIONS AND METHODS FOR TREATING DEPRESSION DISORDERS NOVARTIS AG (CH) 2025-06-12 WO disclosed
EP-4531851-A1 SUBCUTANEOUS ADMINISTRATION OF ONFASPRODIL AND DOSING METHODS FOR USE IN THE TREATMENT OF DEPRESSION DISORDERS Novartis AG (CH) 2025-04-09 EP disclosed
EP-4531851-A1 SUBCUTANEOUS ADMINISTRATION OF ONFASPRODIL AND DOSING METHODS FOR USE IN THE TREATMENT OF DEPRESSION DISORDERS Novartis AG (CH) 2025-04-09 EP disclosed
CN-119654149-A Subcutaneous administration and dosing method of olanzapine for use in the treatment of depressive disorders 诺华股份有限公司 2025-03-18 CN disclosed
WO-2024150146-A1 ENGINEERED KETOREDUCTASE POLYPEPTIDES NOVARTIS AG (CH) 2024-07-18 WO disclosed
WO-2024123935-A2 TREATMENT OR PREVENTION OF DEPRESSIVE DISORDERS THROUGH COMBINATION THERAPY FREEDOM BIOSCIENCES, INC. (US) 2024-06-13 WO disclosed
WO-2023233357-A1 SUBCUTANEOUS ADMINISTRATION OF ONFASPRODIL AND DOSING METHODS FOR USE IN THE TREATMENT OF DEPRESSION DISORDERS NOVARTIS AG (CH) 2023-12-07 WO disclosed
WO-2023233357-A1 SUBCUTANEOUS ADMINISTRATION OF ONFASPRODIL AND DOSING METHODS FOR USE IN THE TREATMENT OF DEPRESSION DISORDERS NOVARTIS AG (CH) 2023-12-07 WO disclosed