SCHEMBL30733142

SCHEMBL30733142

Cc1[nH]c(/C=C2\C(=O)Nc3ccc(F)cc32)c(C)c1C(N)=O

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 2/20 0.82
PRKAA1 Q13131 7/20 0.72
PRKAA2 P54646 6/20 0.72
KDR P35968 10/20 0.68
TLK2 Q86UE8 3/20 0.68
PDGFRB P09619 11/20 0.67
FGFR1 P11362 7/20 0.67
FLT1 P17948 2/20 0.67
HDAC3 O15379 3/20 0.66
HDAC4 P56524 3/20 0.66
HDAC1 Q13547 3/20 0.66
HDAC7 Q8WUI4 3/20 0.66
HDAC2 Q92769 3/20 0.66
HDAC10 Q969S8 3/20 0.66
HDAC11 Q96DB2 3/20 0.66
HDAC8 Q9BY41 3/20 0.66
HDAC6 Q9UBN7 3/20 0.66
HDAC9 Q9UKV0 3/20 0.66
HDAC5 Q9UQL6 3/20 0.66
PLK4 O00444 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29486525 1.00 ALK (0.82) ALKPRKAA1PRKAA2KDRTLK2
SCHEMBL17503076 1.00 ALK (0.82) ALKPRKAA1PRKAA2KDRTLK2
SCHEMBL12329173 1.00 ALK (0.82) ALKPRKAA1PRKAA2KDRTLK2
SCHEMBL859965 0.90 ALK (1.00) ALKPRKAA1PRKAA2KDRTLK2
SCHEMBL859966 0.90 ALK (1.00) ALKPRKAA1PRKAA2KDRTLK2
SCHEMBL8210235 0.90 ALK (0.83) ALKPRKAA1PRKAA2KDRTLK2
SCHEMBL1081676 0.89 ALK (0.82) ALKPRKAA1PRKAA2KDRTLK2
SCHEMBL18814394 0.89 ALK (0.82) ALKPRKAA1PRKAA2KDRTLK2
SCHEMBL21966227 0.88 PRKAA1 (0.80) ALKPRKAA1PRKAA2KDRTLK2
SCHEMBL16085063 0.88 ALK (0.80) ALKPRKAA1PRKAA2KDRTLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117377495-A Non-peptide targeted therapeutic agent and use thereof 克林提克斯医药股份有限公司 2024-01-09 CN disclosed