SCHEMBL30733360

SCHEMBL30733360

C=CC(=O)Nc1cccc(Nc2nc(Nc3ccc(N4CCC(C(C)=O)CC4)cc3OC)ncc2C(F)(F)F)c1

nearest known ligand 0.84

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.84
GAK O14976 1/20 0.84
FES P07332 1/20 0.84
FER P16591 1/20 0.84
ERBB3 P21860 1/20 0.84
TEC P42680 1/20 0.84
CLK1 P49759 1/20 0.84
JAK3 P52333 1/20 0.84
PTK2 Q05397 1/20 0.84
BTK Q06187 1/20 0.84
TNK1 Q13470 1/20 0.84
ALK Q9UM73 1/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Rociletinib SCHEMBL29350136 0.91 EGFR (1.00) EGFRGAKFESFERERBB3
Rociletinib SCHEMBL4177736 0.91 EGFR (1.00) EGFRGAKFESFERERBB3
Rociletinib SCHEMBL29448192 0.91 EGFR (1.00) EGFRGAKFESFERERBB3
SCHEMBL17002256 0.91 EGFR (0.88) EGFRGAKFESFERERBB3
Rociletinib SCHEMBL30101824 0.91 EGFR (0.99) EGFRGAKFESFERERBB3
SCHEMBL2730294 0.91 EGFR (1.00) EGFRGAKFESFERERBB3
SCHEMBL4171719 0.91 EGFR (1.00) EGFRGAKFESFERERBB3
SCHEMBL4165885 0.90 EGFR (1.00) EGFRGAKFESFERERBB3
SCHEMBL18970175 0.90 EGFR (0.86) EGFRGAKFESFERERBB3
SCHEMBL16366037 0.89 EGFR (1.00) EGFRGAKFESFERERBB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117479943-A EGFR inhibitors and PERK activators in combination therapies and use thereof for treating cancer 基因泰克公司 2024-01-30 CN disclosed