SCHEMBL30761111

SCHEMBL30761111

Cc1ccncc1-c1ccnc(C(=O)Nc2ccc(F)cn2)c1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.55
ABL1 P00519 8/20 0.48
CYP1A2 P05177 3/20 0.47
CYP2C9 P11712 3/20 0.47
KCNH2 Q12809 1/20 0.47
CYP3A4 P08684 2/20 0.47
SLC6A3 Q01959 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30761187 0.88 GRM5 (0.60) GRM5CYP1A2CYP2C9KCNH2CYP3A4
SCHEMBL30761151 0.86 GRM5 (0.50) GRM5ABL1CYP1A2CYP2C9KCNH2
SCHEMBL30761114 0.85 GRM5 (0.49) GRM5ABL1CYP1A2CYP2C9KCNH2
SCHEMBL31318893 0.84 ABL1 (0.51) GRM5ABL1
SCHEMBL31318873 0.83 CYP3A4 (0.55) GRM5ABL1CYP1A2CYP2C9CYP3A4
SCHEMBL29236193 0.82 KDM4E (0.50) GRM5ABL1CYP3A4
SCHEMBL31027181 0.82 KDM4E (0.50) GRM5ABL1CYP3A4
SCHEMBL30300046 0.81 ABL1 (0.44) GRM5ABL1
SCHEMBL30761195 0.81 GRM5 (0.52) GRM5ABL1CYP1A2CYP2C9KCNH2
SCHEMBL30761217 0.81 GRM5 (0.52) GRM5CYP1A2CYP2C9KCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024059204-A1 HETEROARYL ANALOGS AS MGLU5 NEGATIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING THE SAME VANDERBILT UNIVERSITY (US) 2024-03-21 WO disclosed