SCHEMBL30763389

SCHEMBL30763389

Clc1cc2c(NCc3cccs3)nc(N3CCNCC3)nc2cn1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 9/20 0.60
HRH1 P35367 1/20 0.60
KHK P50053 2/20 0.50
ALDH1A1 P00352 4/20 0.45
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 2/20 0.45
HPGD P15428 1/20 0.45
HTR3A P46098 1/20 0.43
BRD4 O60885 1/20 0.43
NPC1 O15118 1/20 0.43
HSD17B10 Q99714 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
USP2 O75604 1/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
GLA P06280 1/20 0.43
CYP2C9 P11712 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21686870 1.00 HRH4 (0.60) HRH4HRH1KHKALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL23855480 0.99 HRH4 (0.59) HRH4HRH1KHKALDH1A1CYP1A2
SCHEMBL21686826 0.89 HRH4 (0.75) HRH4HRH1HTR3ABRD4PDE5A
SCHEMBL30763423 0.89 HRH4 (0.75) HRH4HRH1HTR3ABRD4PDE5A
SCHEMBL21686911 0.88 HRH4 (0.62) HRH4HRH1ALDH1A1HTR3ABRD4
SCHEMBL21686942 0.88 HRH4 (0.57) HRH4HRH1KHKALDH1A1CYP1A2
SCHEMBL30763388 0.88 HRH4 (0.57) HRH4HRH1KHKALDH1A1CYP1A2
SCHEMBL30763437 0.87 HRH4 (0.59) HRH4HRH1HTR3ABRD4NPC1
SCHEMBL21687030 0.87 HRH4 (0.59) HRH4HRH1HTR3ABRD4NPC1
SCHEMBL21686914 0.86 HRH4 (0.70) HRH4HRH1HTR3ABRD4PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112739699-B Pyridopyrimidine compounds as histamine H4 receptor inhibitors 费斯制药股份有限公司 2023-11-28 CN disclosed