SCHEMBL30765246

SCHEMBL30765246

Cn1cc(-c2cc3nccc(-c4cncc(S(C)(=O)=O)c4)c3o2)ccc1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.40
PIK3C3 Q8NEB9 1/20 0.36
PIK3CG P48736 4/20 0.36
PIK3CB P42338 3/20 0.36
PIK3CD O00329 2/20 0.36
PIK3CA P42336 2/20 0.36
ADORA2A P29274 3/20 0.34
ADORA1 P30542 3/20 0.34
ADORA2B P29275 2/20 0.34
PI4KA P42356 1/20 0.34
PI4KB Q9UBF8 1/20 0.34
CREBBP Q92793 1/20 0.34
ADORA3 P0DMS8 2/20 0.34
BMPR1B O00238 1/20 0.34
BMPR1A P36894 1/20 0.34
ACVRL1 P37023 1/20 0.34
ACVR1 Q04771 1/20 0.34
DYRK1B Q9Y463 1/20 0.33
DYRK1A Q13627 1/20 0.33
PRKDC P78527 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL725211 0.83 CCNC (0.40) BRD4PIK3C3PIK3CGPIK3CBPIK3CD
SCHEMBL30765349 0.83 BRD4 (0.38) BRD4ADORA2AADORA1ADORA2BCREBBP
SCHEMBL30765399 0.80 BRD4 (0.37) BRD4ADORA2AADORA1ADORA2BCREBBP
SCHEMBL725130 0.80 PIK3C3 (0.36) PIK3C3PIK3CGPIK3CBPIK3CDPIK3CA
SCHEMBL723620 0.79 CYP3A4 (0.38) PIK3C3
SCHEMBL723480 0.78 PIK3C3 (0.39) PIK3C3PIK3CGPIK3CBPIK3CDPIK3CA
SCHEMBL723291 0.78 PIK3C3 (0.36) PIK3C3PIK3CGPIK3CBPIK3CDPIK3CA
SCHEMBL15216703 0.78 PIK3C3 (0.38) BRD4PIK3C3PIK3CGPIK3CBPIK3CD
SCHEMBL27260818 0.77 KCNH2 (0.37) BRD4PIK3CBPIK3CDADORA2AADORA1
SCHEMBL725049 0.77 PIM1 (0.41) BMPR1BBMPR1AACVRL1ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024033280-A1 FUROPYRIDIN AND FUROPYRIMIDIN, INHIBITORS OF PI4K, FOR USE IN THE TREATMENT OF PARASITE INFECTION AND MALARIA MERCK PATENT GMBH (DE) 2024-02-15 WO disclosed