SCHEMBL30775679

SCHEMBL30775679

CC(C)(C)c1cnnc(N)n1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.42
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
HRH4 Q9H3N8 2/20 0.33
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
KDM4E B2RXH2 3/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1605148 1.00 HSD17B10 (0.42) HSD17B10ADORA2AADORA1HRH4HSP90AA1
SCHEMBL12707369 0.88 HSD17B10 (0.34) HSD17B10ADORA2AADORA1
SCHEMBL2652226 0.83 HSP90AA1 (0.38) HSD17B10ADORA2AADORA1HSP90AA1HSP90AB1
SCHEMBL2657204 0.83 HSP90AA1 (0.38) HSD17B10ADORA2AADORA1HSP90AA1HSP90AB1
SCHEMBL2651105 0.83 ADORA2A (0.35) HSD17B10ADORA2AADORA1HSP90AA1HSP90AB1
SCHEMBL30754263 0.77 HSP90AA1 (0.45) HSD17B10ADORA2AADORA1HSP90AA1HSP90AB1
SCHEMBL2651405 0.77 HSP90AA1 (0.45) HSD17B10ADORA2AADORA1HSP90AA1HSP90AB1
SCHEMBL12707361 0.77 ADORA2A (0.32) ADORA2AADORA1
SCHEMBL13172396 0.74 KDM4E (0.31) KDM4E
SCHEMBL278834 0.74 KDM4E (0.31) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4568746-A1 BICYCLIC TETRAHYDROTHIAZEPINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2025-06-18 EP disclosed
CN-119768401-A Bicyclic tetrahydrothiazepine derivatives 豪夫迈·罗氏有限公司 2025-04-04 CN disclosed