SCHEMBL30778358

SCHEMBL30778358

COc1ncc2cc(-c3cnccc3C)[nH]c2c1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
CLK2 P49760 2/20 0.38
CLK3 P49761 2/20 0.38
DYRK1A Q13627 2/20 0.38
ABL1 P00519 2/20 0.38
CHUK O15111 1/20 0.35
PRKD3 O94806 1/20 0.35
PRKCG P05129 1/20 0.35
PRKCB P05771 1/20 0.35
PRKCA P17252 1/20 0.35
CSNK2A2 P19784 1/20 0.35
PRKCH P24723 1/20 0.35
PRKCI P41743 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35
PRKCE Q02156 1/20 0.35
PRKCQ Q04759 1/20 0.35
PRKCZ Q05513 1/20 0.35
PRKCD Q05655 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24753673 1.00 CYP11B1 (0.42) CYP11B1CYP11B2CLK2CLK3DYRK1A
SCHEMBL30059257 0.86 FGFR2 (0.42) KDM5AKDM4CKDM5BTTK
SCHEMBL24753289 0.76 AXL (0.34) CHUKPRKD3PRKCGPRKCBPRKCA
SCHEMBL24753674 0.72 CYP11B1 (0.35) CYP11B1CYP11B2CLK2CLK3DYRK1A
SCHEMBL30056998 0.72 CYP11B1 (0.35) CYP11B1CYP11B2CLK2CLK3DYRK1A
SCHEMBL15036345 0.72 CLK2 (0.40) CYP11B1CYP11B2CLK2CLK3DYRK1A
SCHEMBL24753558 0.71 MAP4K1 (0.40)
SCHEMBL1459164 0.70 CYP19A1 (0.48) CLK2CLK3DYRK1ACHUK
SCHEMBL24754301 0.70
SCHEMBL24754324 0.70 SYK (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117460732-A Pyrrolopyridone compounds, preparation method and application thereof 杭州中美华东制药有限公司 2024-01-26 CN disclosed