SCHEMBL30779604

SCHEMBL30779604

CC(C)c1cc(C(=O)N(c2ccccc2F)C(C)C)c(O)cc1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 14/20 0.52
HSP90AB1 P08238 2/20 0.45
MET P08581 1/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP2B6 P20813 1/20 0.44
HDAC3 O15379 3/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC7 Q8WUI4 2/20 0.41
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP3A5 P20815 1/20 0.39
CYP3A7 P24462 1/20 0.39
CYP3A43 Q9HB55 1/20 0.39
HDAC2 Q92769 2/20 0.38
HDAC11 Q96DB2 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
HDAC5 Q9UQL6 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21644697 1.00 HSP90AA1 (0.52) HSP90AA1HSP90AB1METCYP3A4CYP2C9
SCHEMBL21644514 0.86 HSP90AA1 (0.56) HSP90AA1HSP90AB1METCYP3A4CYP2C9
SCHEMBL30779551 0.86 HSP90AA1 (0.56) HSP90AA1HSP90AB1METCYP3A4CYP2C9
SCHEMBL21644574 0.82 CYP3A4 (0.58) HSP90AA1HSP90AB1METCYP3A4CYP2C9
SCHEMBL30779627 0.82 CYP3A4 (0.58) HSP90AA1HSP90AB1METCYP3A4CYP2C9
SCHEMBL21644597 0.81 HSP90AA1 (0.60) HSP90AA1HSP90AB1METCYP3A4CYP2C9
SCHEMBL21644682 0.81 HSP90AA1 (0.51) HSP90AA1HSP90AB1METCYP3A4CYP2C9
SCHEMBL30779629 0.81 HSP90AA1 (0.51) HSP90AA1HSP90AB1METCYP3A4CYP2C9
SCHEMBL21644563 0.79 HSP90AA1 (0.48) HSP90AA1HSP90AB1METCYP3A4CYP2C9
SCHEMBL21644591 0.79 CYP3A4 (0.48) HSP90AA1HSP90AB1METCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111164074-B Heat shock protein 90 inhibitors 台北医学大学 2024-02-02 CN disclosed